General Information of Drug (ID: DM942HP)

Drug Name
Brivanib
Synonyms
Brivanib; 649735-46-6; BMS-540215; Brivanib (BMS-540215); BMS 540215; UNII-DDU33B674I; Brivanib [USAN]; BMS540215; DDU33B674I; CHEMBL377300; (2R)-1-[4-(4-Fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]propanol; Brivanib (USAN); (2R)-1-[4-[(4-FLUORO-2-METHYL-1H-INDOL-5-YL)OXY]-5-METHYL-PYRROLO[2,1-F][1,2,4]TRIAZIN-6-YL]OXYPROPAN-2-OL; (2R)-1-({4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl}oxy)propan-2-ol
Indication
Disease Entry ICD 11 Status REF
Breast cancer 2C60-2C65 Phase 3 [1]
Liver cancer 2C12 Phase 3 [1]
Drug Type
Small molecular drug
Structure
3D MOL 2D MOL
#Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 370.4
Logarithm of the Partition Coefficient (xlogp) 3
Rotatable Bond Count (rotbonds) 5
Hydrogen Bond Donor Count (hbonddonor) 2
Hydrogen Bond Acceptor Count (hbondacc) 6
Chemical Identifiers
Formula
C19H19FN4O3
IUPAC Name
(2R)-1-[4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl]oxypropan-2-ol
Canonical SMILES
CC1=CC2=C(N1)C=CC(=C2F)OC3=NC=NN4C3=C(C(=C4)OC[C@@H](C)O)C
InChI
InChI=1S/C19H19FN4O3/c1-10-6-13-14(23-10)4-5-15(17(13)20)27-19-18-12(3)16(26-8-11(2)25)7-24(18)22-9-21-19/h4-7,9,11,23,25H,8H2,1-3H3/t11-/m1/s1
InChIKey
WCWUXEGQKLTGDX-LLVKDONJSA-N
Cross-matching ID
PubChem CID
11234052
ChEBI ID
CHEBI:94562
CAS Number
649735-46-6
UNII
DDU33B674I
DrugBank ID
DB11958
TTD ID
D0HS5V
Combinatorial Drugs (CBD) Click to Jump to the Detailed CBD Information of This Drug
Repurposed Drugs (RPD) Click to Jump to the Detailed RPD Information of This Drug

Molecular Interaction Atlas of This Drug


Drug Therapeutic Target (DTT)
DTT Name DTT ID UniProt ID MOA REF
Vascular endothelial growth factor receptor 2 (KDR) TTUTJGQ VGFR2_HUMAN Modulator [2]
Molecular Interaction Atlas (MIA) Jump to Detail Molecular Interaction Atlas of This Drug

Molecular Expression Atlas of This Drug

The Studied Disease Breast cancer
ICD Disease Classification 2C60-2C65
Molecule Name Molecule Type Gene Name p-value Fold-Change Z-score
Vascular endothelial growth factor receptor 2 (KDR) DTT KDR 1.98E-01 0.11 0.2
Molecular Expression Atlas (MEA) Jump to Detail Molecular Expression Atlas of This Drug

Experimental Cancer Drug Sensitivity Information

Cancer Drug Sensitivity Data Curated from 50 Cell Line(s) in Bone Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
RPMI-3460/CS1 GDSC1 5.876 8.7005 3.2521 4.1878
EW-13 GDSC1 1.5507 4.1344 1.3467 35.7989
H-EMC-SS GDSC1 2.1888 7.1969 0.8688 33.9988
ES1 GDSC1 2.7751 6.3583 1.8397 25.6225
U2OS CTRP2 3.0037 4.9254 2.9513 20.4348
NOS-1 [Human HNSCC] GDSC1 3.5931 7.8175 1.9349 21.1011
CADO-ES1 GDSC1 3.7132 6.1628 2.8554 13.9589
MHH-ES-1 GDSC1 4.2392 7.2361 2.7953 12.2911
SK-PN-DW GDSC1 4.2434 7.0986 2.8676 11.7209
U2OS GDSC1 4.255 8.0446 2.4045 15.1499
EW-1 GDSC1 4.3721 7.5007 2.7742 11.9634
TC71 CTRP2 4.3768 8.7276 3.1463 15.8196
EW-3 GDSC1 4.4059 8.796 2.1545 16.3589
ES7 GDSC1 4.4775 8.1656 2.5282 13.4311
SK-ES-1 GDSC1 4.4824 9.0837 2.0734 16.6342
EW-7 GDSC1 4.6886 7.0582 3.2461 7.2405
HOS GDSC1 4.7542 8.3936 2.6342 11.6979
SJSA-1 GDSC1 4.7764 7.7414 2.9746 9.0571
NY GDSC1 4.8141 7.7213 3.013 8.645
ES8 GDSC1 4.8702 8.5621 2.6396 11.2805
CHSA8926 GDSC1 4.9271 7.4838 3.2126 6.7767
A-673 GDSC1 5.0515 10.7544 1.6916 17.144
EW-22 GDSC1 5.1391 10.1079 2.0785 14.378
EW-16 GDSC1 5.1449 8.0508 3.0908 7.0818
HuO9 GDSC1 5.1451 11.9409 1.1749 19.826
EW-18 GDSC1 5.1472 8.7567 2.7491 9.621
ES4 GDSC1 5.1538 8.3412 2.9563 8.0639
SK-N-MC CTRP2 5.1912 7.8566 4.3565 8.9336
G-292 clone A141B1 GDSC1 5.2732 9.2598 2.5939 10.3823
MHH-ES-1 CTRP2 5.2907 7.9804 4.3939 8.5438
TC-71 GDSC1 5.3135 8.938 2.7789 8.9244
CAL-78 CTRP2 5.3395 7.3052 4.7608 6.9303
HuO-3N1 GDSC1 5.3844 11.3349 1.6567 16.2997
EW-24 GDSC1 5.4048 7.1573 3.6726 2.2822
CAL-72 GDSC1 5.4126 7.2761 3.6242 2.5872
A-673 CTRP2 5.4999 9.1773 4.0039 9.6874
ES6 GDSC1 5.5105 8.6947 3.0291 6.5779
SK-ES-1 CTRP2 5.6231 7.8437 4.7733 6.2157
ES5 GDSC1 5.8008 8.4209 3.3342 3.7829
CAL-78 GDSC1 6.0692 10.2112 2.6748 7.7245
HOS CTRP2 6.1567 9.01 4.6541 5.6307
G-292 clone A141B1 CTRP2 6.4394 10.8629 3.9559 8.0392
SJSA-1 CTRP2 6.5266 8.7666 5.0613 3.2894
SaOS-2 CTRP2 6.6062 7.95 5.5092 1.3681
SaOS-2 GDSC1 6.6344 12.2081 2.0991 10.1723
MG-63 GDSC1 6.9659 13.4648 1.7214 11.6804
SW1353 CTRP2 7.1103 9.277 5.2064 1.9192
Hs 822.T CTRP2 7.2814 8.2433 5.7282 0.168
Hs 888.T CTRP2 7.7656 9.9928 5.253 1.1352
MG-63 CTRP2 8.0534 10.5005 5.1843 1.1309
⏷ Show the Full List of 50 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 287 Cell Line(s) in Haematopoietic And Lymphoid Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MEC1 CTRP2 3.649 6.0851 3.419 16.764
JK1 CTRP2 4.9732 8.3733 3.8999 11.3186
JM1 CTRP2 4.6426 7.5801 3.9325 12.0145
JM1 GDSC1 4.7612 8.7433 2.4658 12.9091
DND-41 CTRP2 0.2465 1.3548 0.2465 38.6265
EoL-1 GDSC1 0.7762 2.4893 0.7599 44.392
EoL-1 CTRP2 1.3561 2.5055 1.3559 31.2349
SUP-M2 CTRP2 1.4112 2.1883 1.4112 30.8668
KG-1 GDSC1 1.4955 4.9508 1.0452 37.6262
SU-DHL-1 CTRP2 1.5506 3.2385 1.5462 29.9532
MV4-11 CTRP2 1.867 3.3922 1.8636 27.8417
SIG-M5 GDSC1 1.8818 4.3209 1.6592 31.8705
SK-MM-2 CTRP2 1.985 5.4366 1.7642 27.7958
KMS-12-BM CTRP2 2.0229 4.8168 1.9197 27.141
697 GDSC1 2.105 6.2408 1.2017 32.9629
CML-T1 CTRP2 2.4244 4.4887 2.3853 24.2484
CTB-1 GDSC1 2.4491 5.7599 1.7627 27.8647
WIL2 NS GDSC1 2.4608 6.0875 1.6366 28.557
SU-DHL-5 GDSC1 2.4616 5.5506 1.8614 27.1809
Karpas-231 GDSC1 2.5732 6.1436 1.7284 27.3887
HAL-01 GDSC1 2.6118 7.2371 1.2744 29.7474
H9 GDSC1 2.6297 6.8296 1.4796 28.5406
SU-DHL-10 GDSC1 2.638 6.4362 1.6657 27.4168
OPM-2 GDSC1 2.6736 4.8227 2.3651 22.665
WSU-DLCL2 CTRP2 2.7111 5.4075 2.5586 22.7301
MV4-11 GDSC1 2.72 7.2756 1.3636 28.7063
VAL GDSC1 2.8375 6.2932 1.9321 24.7074
KE-97 CTRP2 2.8746 5.5932 2.697 21.73
MN-60 GDSC1 2.9337 6.8099 1.7917 25.1125
KE-37 GDSC1 3.0118 6.4525 2.0347 23.1498
BL-70 CTRP2 3.012 4.7727 2.9763 20.3225
RPMI-8866 GDSC1 3.0325 6.3762 2.0905 22.6721
MOLM-13 CTRP2 3.1111 5.5345 2.9666 20.0393
OCI-AML-2 GDSC1 3.1223 5.5886 2.5354 19.1049
RCH-ACV GDSC1 3.1637 7.0957 1.8818 23.4113
RCH-ACV CTRP2 3.1951 6.1011 2.9192 19.9484
TUR GDSC1 3.2048 6.8293 2.0482 22.1191
Raji CTRP2 3.2152 5.5281 3.0809 19.3103
HC-1 GDSC1 3.2381 8.1139 1.4612 25.617
DB CTRP2 3.2848 6.1575 3.0012 19.3799
GA-10 GDSC1 3.3093 6.3649 2.3695 19.3917
SU-DHL-16 GDSC1 3.3277 5.5663 2.7553 16.4882
BC-1 GDSC1 3.3332 5.929 2.5962 17.633
Ku812 GDSC1 3.3537 9.3999 0.9369 27.8503
Reh GDSC1 3.3732 7.2906 1.9881 21.734
A3/Kawakami GDSC1 3.3899 6.3937 2.4345 18.5472
SU-DHL-8 CTRP2 3.4081 7.753 2.5706 20.6211
SU-DHL-10 CTRP2 3.4231 7.4013 2.7253 19.9974
NALM-6 GDSC1 3.4291 8.504 1.4471 24.8269
SU-DHL-8 GDSC1 3.4732 7.9051 1.7818 22.617
A3/Kawakami CTRP2 3.4877 6.1566 3.2227 17.9635
P30/OHK GDSC1 3.5544 7.1903 2.2068 19.4258
M-07e CTRP2 3.5964 6.8198 3.1271 17.995
KMS-28BM CTRP2 3.637 6.7712 3.188 17.65
SR CTRP2 3.6496 6.9873 3.124 17.8535
IM-9 GDSC1 3.7067 6.3725 2.7476 14.8049
EM-2 CTRP2 3.7069 6.5182 3.3499 16.844
LAMA-84 GDSC1 3.7238 6.726 2.5911 15.9077
OCI-Ly19 GDSC1 3.7292 8.0288 1.9539 20.3902
697 CTRP2 3.7342 6.7114 3.314 16.8977
KMS-26 CTRP2 3.743 6.2258 3.4811 16.2551
Sc-1 GDSC1 3.7542 7.6698 2.1541 18.9287
HEL CTRP2 3.7765 7.1633 3.194 17.2292
Mino CTRP2 3.8273 6.7427 3.4036 16.2936
RPMI-8402 CTRP2 3.8664 6.6946 3.4628 15.9593
DEL CTRP2 3.8718 8.0412 2.9372 17.9523
NU-DUL-1 GDSC1 3.8804 7.3219 2.4398 16.368
Daudi CTRP2 3.8847 6.2761 3.6203 15.3222
MY-M12 GDSC1 3.8888 8.8759 1.6746 21.5081
KMS-34 CTRP2 3.8994 5.7915 3.7674 14.7468
RPMI-6666 GDSC1 3.906 7.253 2.4968 15.8441
NALM-6 CTRP2 3.9118 6.5911 3.5477 15.5105
NCO2 CTRP2 3.9245 5.9084 3.7666 14.6721
Jurkat CTRP2 3.9526 7.8718 3.0931 17.1321
U-937 CTRP2 3.966 7.1428 3.404 15.8981
Raji GDSC1 3.9723 7.958 2.2049 17.6753
JSC-1 GDSC1 3.9858 6.5739 2.9048 12.4343
KMS-11 CTRP2 4.0022 7.6013 3.2583 16.3584
BALL-1 GDSC1 4.0044 7.7798 2.3217 16.7199
GDM-1 GDSC1 4.0423 7.0505 2.7182 13.6379
P32/ISH GDSC1 4.052 8.262 2.1226 17.9279
KMS-12-BM GDSC1 4.0661 10.9445 0.7952 25.589
NB4 GDSC1 4.076 7.2385 2.654 13.991
KOPN-8 GDSC1 4.0808 9.1876 1.6854 20.6704
KCL-22 GDSC1 4.0852 9.2727 1.6465 20.8918
SIG-M5 CTRP2 4.0921 6.496 3.7753 14.1377
MC116 CTRP2 4.1108 7.2941 3.498 15.1362
Jurkat GDSC1 4.1363 8.9167 1.868 19.297
MOLM-13 GDSC1 4.142 8.7044 1.979 18.5459
K-562 GDSC1 4.1621 7.8304 2.4328 15.2986
Ri-1 CTRP2 4.173 8.4147 3.0832 16.5893
KE-37 CTRP2 4.1735 6.0372 4.0046 13.0546
OCI-AML-5 GDSC1 4.1961 7.7528 2.5005 14.6718
CESS GDSC1 4.1986 8.7669 1.9958 18.2153
QIMR-WIL GDSC1 4.2023 7.6895 2.5375 14.3748
Ki-JK CTRP2 4.2119 6.8122 3.7926 13.7278
KMS-21-BM CTRP2 4.2309 5.828 4.12 12.4653
SUP-T1 GDSC1 4.247 8.4361 2.2021 16.6217
Ramos.2G6.4C10 GDSC1 4.2599 7.6478 2.607 13.6396
JVM-3 CTRP2 4.28 6.9581 3.8102 13.469
PL-21 GDSC1 4.2959 8.6614 2.1305 16.9329
Karpas-620 CTRP2 4.3328 6.3211 4.0942 12.2498
NU-DUL-1 CTRP2 4.3532 7.0032 3.8705 13.0345
BC-3 GDSC1 4.3532 7.8503 2.5838 13.4676
THP-1 GDSC1 4.3542 8.2007 2.4094 14.7459
HEL GDSC1 4.36 7.1415 2.9438 10.7041
RL CTRP2 4.3611 6.7546 3.9741 12.6175
DoHH2 GDSC1 4.4017 8.258 2.42 14.4944
CA46 CTRP2 4.4171 7.4159 3.7696 13.2513
MOLT-4 GDSC1 4.4367 8.7039 2.2258 15.7512
JURL-MK1 CTRP2 4.4623 6.7227 4.0946 11.8736
AML-193 CTRP2 4.4673 7.3767 3.8385 12.8475
SUP-M2 GDSC1 4.4756 7.7907 2.7138 12.0524
RPMI-8402 GDSC1 4.491 7.5943 2.8245 11.1575
P12-Ichikawa CTRP2 4.5232 7.5545 3.8206 12.769
P12-Ichikawa GDSC1 4.5293 7.198 3.0529 9.2649
RS4;11 GDSC1 4.5317 9.8868 1.7123 18.8025
Ku812 CTRP2 4.5445 6.8965 4.1158 11.5626
HH [Human lymphoma] GDSC1 4.5959 8.3562 2.5283 13.0151
Peer CTRP2 4.5967 7.2184 4.0401 11.7129
KMM-1 CTRP2 4.6077 6.9977 4.1424 11.2861
OCI-Ly3 CTRP2 4.6169 7.2486 4.0485 11.6259
KCL-22 CTRP2 4.6277 7.269 4.0511 11.5868
Jiyoye GDSC1 4.631 8.0753 2.6962 11.6474
MC116 GDSC1 4.6504 6.6556 3.4163 6.0363
SUP-B15 GDSC1 4.6633 6.6039 3.4515 5.7226
MOLT-16 GDSC1 4.6785 7.1834 3.1764 7.8128
SU-DHL-4 CTRP2 4.6868 8.1473 3.7225 12.7389
OCI-M1 GDSC1 4.7045 8.5928 2.4963 12.8779
TF-1 CTRP2 4.7072 8.4667 3.5951 13.2007
Mono-Mac-6 GDSC1 4.7261 8.3631 2.6275 11.8412
RPMI-6666 CTRP2 4.7469 7.6762 3.9965 11.4906
PF-382 CTRP2 4.7733 8.0701 3.8444 12.0328
NK-92MI GDSC1 4.7781 10.4182 1.6451 18.3473
L-363 GDSC1 4.8091 7.0722 3.3287 6.2324
BE-13 GDSC1 4.8157 8.2907 2.7325 10.7655
ML-2 GDSC1 4.8163 7.5759 3.0863 8.0764
HH [Human lymphoma] CTRP2 4.8223 8.8861 3.5101 13.265
MOLT-13 GDSC1 4.8377 8.3828 2.7037 10.9098
L-540 GDSC1 4.8503 9.6729 2.073 15.355
L-428 CTRP2 4.853 7.7828 4.0557 10.9842
Mono-Mac-6 CTRP2 4.8758 11.8066 2.1396 18.558
LP-1 GDSC1 4.8931 8.2423 2.815 9.9006
GA-10 CTRP2 4.9085 6.5657 4.6316 8.5743
HEL 92.1.7 CTRP2 4.9162 7.8865 4.0714 10.7628
PF-382 GDSC1 4.9207 8.5762 2.6709 10.8892
LAMA-84 CTRP2 4.9276 7.6905 4.1726 10.3272
K-562 CTRP2 4.9287 7.6 4.2148 10.1551
RPMI-8226 GDSC1 4.9425 8.4026 2.7728 10.0632
JVM-2 CTRP2 4.947 7.7391 4.1699 10.2893
A4/Fukuda GDSC1 4.9478 8.1746 2.8891 9.1744
SKM-1 GDSC1 4.9509 8.5666 2.6983 10.5913
Farage GDSC1 4.952 8.2469 2.8566 9.4059
BV-173 GDSC1 4.9559 11.7412 1.1265 20.7091
F-36P CTRP2 4.9634 9.4267 3.3853 13.4404
SUP-HD1 GDSC1 4.9641 9.8578 2.0693 15.0034
MOLT-16 CTRP2 4.9644 6.6197 4.6706 8.2685
MJ CTRP2 4.967 10.2811 2.9726 15.1033
BL-41 GDSC1 4.9683 7.591 3.1897 6.8324
EM-2 GDSC1 4.9736 7.3223 3.324 5.7957
Namalwa CTRP2 4.9773 7.8625 4.1432 10.3212
Daudi GDSC1 5.023 8.1667 2.9479 8.5051
L-540 CTRP2 5.0247 7.1025 4.5339 8.6379
HL-60 GDSC1 5.0269 9.4826 2.303 13.2011
JURL-MK1 GDSC1 5.0343 7.1974 3.4258 4.8645
SU-DHL-6 GDSC1 5.0605 8.4675 2.8279 9.2938
ALL-SIL CTRP2 5.0621 6.3193 4.8865 7.1741
CA46 GDSC1 5.0711 8.8168 2.6642 10.4731
THP-1 CTRP2 5.0913 8.0564 4.1648 9.9553
Granta-519 GDSC1 5.1066 8.7493 2.7232 9.9319
HT GDSC1 5.1154 8.9694 2.6218 10.6488
ALL-PO GDSC1 5.1231 7.9412 3.1287 6.8582
HuNS1 CTRP2 5.1258 8.7734 3.855 11.1419
JeKo-1 CTRP2 5.1308 7.9916 4.2338 9.5791
GR-ST GDSC1 5.138 10.3985 1.934 15.3323
U-698-M GDSC1 5.185 9.4913 2.4165 11.9111
P3HR-1 CTRP2 5.1905 9.7354 3.4466 12.6731
SU-DHL-6 CTRP2 5.2415 8.6387 4.0296 10.1566
BV-173 CTRP2 5.2923 7.7369 4.5115 8.0587
CTV-1 GDSC1 5.2956 7.7988 3.3125 5.0427
ROS-50 GDSC1 5.3166 9.8175 2.3525 11.964
LC4-1 GDSC1 5.3231 7.9606 3.254 5.4036
Hs 445 GDSC1 5.3308 6.933 3.7304 2.0387
L-1236 GDSC1 5.3347 8.6815 2.9175 7.8501
MOLP-8 GDSC1 5.345 9.6683 2.446 11.2261
EB1 CTRP2 5.3495 7.1373 4.8484 6.5518
DB GDSC1 5.3569 8.94 2.8081 8.5909
MEG-01 GDSC1 5.3611 11.9628 1.3292 18.2868
TK [Human B-cell lymphoma] GDSC1 5.3709 8.0693 3.2337 5.4346
ALL-SIL GDSC1 5.386 12.7157 0.9755 20.1132
YT GDSC1 5.4031 7.837 3.3629 4.424
L-428 GDSC1 5.4292 7.5274 3.5209 3.2556
NOMO-1 GDSC1 5.4513 10.4841 2.1238 13.122
SK-MM-2 GDSC1 5.4545 8.1388 3.2546 5.0828
Pfeiffer CTRP2 5.4635 6.1325 5.3844 4.1504
CCRF-CEM GDSC1 5.468 12.6336 1.0783 19.3229
ME1 GDSC1 5.4906 6.9475 3.8078 1.3126
KMS-11 GDSC1 5.4931 10.4928 2.1498 12.8259
LP-1 CTRP2 5.4955 7.6467 4.7498 6.6026
SCC-3 GDSC1 5.5029 10.2917 2.2549 12.0898
P31/FUJ CTRP2 5.5501 9.0366 4.1187 9.1007
MOTN-1 CTRP2 5.5602 7.3724 4.9436 5.6553
MHH-PREB-1 GDSC1 5.5604 8.4297 3.1856 5.3306
MOLM-16 CTRP2 5.5794 8.7367 4.2934 8.3092
KM-H2 CTRP2 5.5909 7.9911 4.6713 6.7109
ARH-77 GDSC1 5.5924 8.6935 3.0825 5.993
A4/Fukuda CTRP2 5.5979 7.2468 5.0399 5.1711
EJM GDSC1 5.6214 9.0068 2.9537 6.846
U266B1 GDSC1 5.6334 7.5583 3.6218 2.2113
RC-K8 GDSC1 5.6491 7.7113 3.5637 2.5527
Hs 611.T CTRP2 5.6592 6.7748 5.3236 3.8654
SUP-T11 CTRP2 5.6735 6.786 5.3325 3.7947
Karpas-45 GDSC1 5.6764 9.415 2.7964 7.8324
EHEB GDSC1 5.6793 8.3875 3.2781 4.4143
KMOE-2 GDSC1 5.699 9.5351 2.7543 8.0741
KYO-1 CTRP2 5.6996 8.6737 4.4324 7.4716
KMS-18 CTRP2 5.7113 8.6201 4.4695 7.2921
NKM-1 GDSC1 5.7142 9.5794 2.7433 8.1131
Karpas-422 GDSC1 5.7153 9.2725 2.8892 7.076
DND-41 GDSC1 5.7171 11.1844 1.9725 13.3409
HDLM-2 GDSC1 5.7392 10.5713 2.285 11.2221
Karpas-620 GDSC1 5.7626 9.5491 2.7894 7.6666
EHEB CTRP2 5.7834 8.5616 4.5622 6.7531
MOLT-3 CTRP2 5.8094 6.6677 5.5203 2.7027
KY821 GDSC1 5.8121 9.1866 2.9909 6.1295
Karpas-422 CTRP2 5.8237 7.2752 5.2367 3.8465
Kasumi-2 CTRP2 5.8266 8.6549 4.5535 6.7002
NCI-H929 CTRP2 5.8379 8.1407 4.8195 5.5614
Kasumi-1 CTRP2 5.8424 7.8821 4.9522 4.9962
ST486 GDSC1 5.848 9.1996 3.0071 5.9339
TALL-1 [Human adult T-ALL] CTRP2 5.8679 9.741 4.047 8.7402
RS4;11 CTRP2 5.9066 8.2868 4.8063 5.4763
KHM-1B CTRP2 5.9259 7.4354 5.2479 3.5841
Ci-1 CTRP2 5.9289 7.0627 5.4361 2.789
AMO1 GDSC1 5.9369 7.2392 3.892 0.4704
JJN-3 CTRP2 5.9426 9.6581 4.1521 8.1509
HT CTRP2 5.9468 6.9753 5.4953 2.5037
DG-75 GDSC1 5.9634 9.7431 2.8266 6.9261
L-363 CTRP2 5.9832 9.3609 4.3349 7.3041
MHH-CALL-3 CTRP2 5.99 8.1364 4.9527 4.6947
AMO1 CTRP2 5.9903 9.0303 4.5062 6.5707
HD-MY-Z CTRP2 6.0033 9.6174 4.2235 7.7322
OCI-Ly10 CTRP2 6.0418 8.457 4.8359 5.0845
P31/FUJ GDSC1 6.0493 7.265 3.9264 0.2983
JVM-2 GDSC1 6.054 8.9741 3.2315 3.9814
OCI-M1 CTRP2 6.0551 7.2791 5.4359 2.5373
MOLM-6 CTRP2 6.0905 8.0447 5.0824 3.9557
Karpas-299 GDSC1 6.1082 11.8724 1.9117 12.6533
SU-DHL-1 GDSC1 6.1132 11.6036 2.044 11.8052
KO52 CTRP2 6.136 6.967 5.6571 1.4596
ATN-1 GDSC1 6.1571 10.2781 2.6989 7.3573
KMS-27 CTRP2 6.1599 8.4499 4.9365 4.4388
SU-DHL-4 GDSC1 6.1689 7.619 3.8447 0.4877
CMK CTRP2 6.1891 7.8882 5.2401 3.1114
WSU-DLCL2 GDSC1 6.1999 7.3184 3.9628 0.1571
SET-2 CTRP2 6.2087 7.4637 5.4666 2.1297
EJM CTRP2 6.2126 7.5567 5.4235 2.3027
EB2 GDSC1 6.2325 8.6433 3.4692 2.2135
U266B1 CTRP2 6.2335 10.7163 3.8642 8.7978
RL GDSC1 6.2363 7.508 3.9103 0.2601
SUP-B15 CTRP2 6.2379 7.5709 5.4358 2.2081
NU-DHL-1 CTRP2 6.2507 7.8994 5.2827 2.8252
JVM-3 GDSC1 6.2526 8.0355 3.7228 0.8983
ME1 CTRP2 6.2577 9.6164 4.4329 6.3725
HL-60 CTRP2 6.2629 7.7158 5.3831 2.3854
VL51 GDSC1 6.2825 11.6376 2.1406 10.7568
Mono-Mac-1 CTRP2 6.294 8.2837 5.1253 3.4074
MLMA GDSC1 6.3002 7.8904 3.7971 0.5696
Granta-519 CTRP2 6.3011 8.5976 4.9749 4.0236
MM1.S CTRP2 6.3684 7.6332 5.5011 1.7291
HDLM-2 CTRP2 6.4393 8.1773 5.2864 2.4999
KM-H2 GDSC1 6.4587 7.813 3.8851 0.2369
OCI-AML-3 GDSC1 6.4664 13.6429 1.3049 15.2695
Loucy GDSC1 6.5021 7.8502 3.8879 0.2165
MOLP-8 CTRP2 6.5595 8.1229 5.3968 1.8738
WSU-NHL GDSC1 6.7914 8.2987 3.8371 0.2312
SUP-HD1 CTRP2 6.8226 8.6971 5.2969 1.9191
SR GDSC1 6.8438 8.7113 3.7112 0.533
HPB-ALL CTRP2 6.861 8.4754 5.4232 1.3925
MOLP-2 CTRP2 7.0386 9.1987 5.1987 2.032
KMS-20 CTRP2 7.058 35.9676 -8.0811 34.7287
MHH-CALL-4 CTRP2 7.1546 9.151 5.2897 1.5634
MOLT-13 CTRP2 8.2119 9.6817 5.5678 0.1711
JJN-3 GDSC1 8.4329 17.1366 0.9303 12.74
OCI-Ly19 CTRP2 8.7866 10.3986 5.5272 0.115
DEL GDSC1 8.9157 18.7147 0.4983 13.8019
OCI-AML-5 CTRP2 10.0667 18.764 2.6422 7.9327
⏷ Show the Full List of 287 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 48 Cell Line(s) in Oesophagus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TE8 CTRP2 6.2817 8.2808 5.1173 3.4624
TE15 CTRP2 6.7358 8.4295 5.367 1.7566
KYSE-510 GDSC1 4.3251 7.8452 2.5629 13.7261
TE-8 GDSC1 4.6083 7.5823 2.9239 9.9947
KYSE-150 GDSC1 4.651 8.6326 2.4343 13.5102
TE-15 GDSC1 4.7281 7.5874 3.0141 8.9086
COLO 680N GDSC1 4.8447 7.0497 3.3653 5.8463
KYSE-270 GDSC1 4.9334 8.8359 2.5521 11.7209
TE-6 GDSC1 5.0912 11.2088 1.4967 18.1862
TE-10 GDSC1 5.3326 10.6512 1.955 14.5883
TE-9 GDSC1 5.333 8.4362 3.0342 6.9951
EC-GI-10 GDSC1 5.3967 10.5033 2.0747 13.6103
KYSE-450 GDSC1 5.4579 8.1421 3.2552 5.0705
KYSE-140 GDSC1 5.5372 9.0201 2.8921 7.5012
KYSE-410 GDSC1 5.5685 8.6327 3.0958 5.9547
TE-5 GDSC1 5.6762 8.1279 3.394 3.6246
TE-4 GDSC1 5.69 8.1152 3.4077 3.5053
KYSE-520 GDSC1 5.7416 9.3643 2.863 7.1983
KYSE-410 CTRP2 5.7805 8.373 4.6535 6.3766
T.T GDSC1 5.7989 9.2369 2.9592 6.3821
OE19 GDSC1 5.9578 7.4088 3.837 0.6656
KYSE-70 GDSC1 5.9891 10.6191 2.4309 9.5802
TE-5 CTRP2 6.0805 7.5755 5.3087 3.0235
TE-11 CTRP2 6.2475 8.5532 4.955 4.2017
KYSE-510 CTRP2 6.2941 10.5221 4.0101 8.0765
KYSE-520 CTRP2 6.2944 7.9344 5.2988 2.6832
TE-11 GDSC1 6.2977 11.3676 2.2782 9.8305
OE21 CTRP2 6.2992 7.6096 5.4627 1.9951
TE-6 CTRP2 6.3222 8.4252 5.0768 3.5615
KYSE-30 CTRP2 6.3519 11.446 3.5954 9.6945
KYSE-180 CTRP2 6.4207 9.2557 4.7405 4.796
TE-10 CTRP2 6.4224 8.1926 5.2667 2.6076
KYSE-70 CTRP2 6.4451 8.1956 5.2817 2.5105
OE21 GDSC1 6.5293 9.8053 3.1279 3.8006
TE-14 CTRP2 6.5522 10.0391 4.4529 5.7709
OE33 GDSC1 6.6436 10.3365 2.958 4.6639
TE-1 GDSC1 6.722 10.7895 2.8015 5.5107
TE-1 CTRP2 6.7957 10.4727 4.4209 5.5028
KYSE-150 CTRP2 6.8089 9.7251 4.7957 3.9441
COLO 680N CTRP2 6.8128 10.0317 4.6492 4.5368
TE-4 CTRP2 6.8327 8.7736 5.2675 2.0207
TE-9 CTRP2 7.0111 11.3192 4.1628 6.2232
KYSE-140 CTRP2 7.0368 9.3148 5.1437 2.2445
KYSE-180 GDSC1 7.4272 14.8706 1.3564 12.6766
OE33 CTRP2 7.4666 10.1152 5.0365 2.1522
EC-GI-10 CTRP2 7.7777 11.7589 4.4701 3.9234
KYSE-450 CTRP2 10.5296 25.7086 -0.3473 16.685
OE19 CTRP2 12.2692 22.9022 2.0638 7.4671
⏷ Show the Full List of 48 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 67 Cell Line(s) in Pancreas Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
N2a-PK1 CTRP2 7.0897 11.359 4.1998 5.9502
HPAC CTRP2 3.6015 7.3894 2.92 18.7603
SUIT-2 GDSC1 4.9178 7.5282 3.1842 7.0207
Panc 03.27 GDSC1 4.9229 7.4204 3.2405 6.5759
KP-1N GDSC1 5.0594 9.862 2.1399 14.2185
MZ-PC-1 GDSC1 5.0788 7.4582 3.3309 5.458
KP-2 CTRP2 5.1571 8.1789 4.1704 9.7752
SU.86.86 GDSC1 5.2468 7.1001 3.607 3.0384
Panc 04.03 GDSC1 5.3279 8.2298 3.1294 6.307
DAN-G GDSC1 5.3497 8.0464 3.2308 5.5078
QGP-1 GDSC1 5.3999 8.4859 3.0552 6.667
MIA PaCa-2 GDSC1 5.4831 8.4779 3.1137 6.0326
HuP-T3 GDSC1 5.546 8.0005 3.375 4.023
PaTu 8988s CTRP2 5.5823 9.0986 4.117 9.039
PL4 GDSC1 5.5997 7.8762 3.4629 3.3096
Capan-1 GDSC1 5.668 7.8946 3.4935 2.9756
PaTu 8988t GDSC1 5.7875 8.5318 3.2766 4.1993
Panc 10.05 GDSC1 5.8747 9.4341 2.9149 6.5172
HPAF-II GDSC1 5.8797 9.4172 2.9259 6.4287
MIA PaCa-2 CTRP2 5.9064 8.676 4.6119 6.2929
KP-4 GDSC1 5.9394 8.3201 3.4555 2.7437
YAPC GDSC1 5.9427 8.5825 3.3426 3.46
Panc 08.13 GDSC1 5.9519 10.561 2.4339 9.6543
HuP-T4 GDSC1 5.9586 9.1764 3.085 5.1547
KP-4 CTRP2 5.9964 8.8275 4.6126 6.1115
Hs 766T GDSC1 5.9992 8.0855 3.5859 1.8727
QGP-1 CTRP2 6.0238 8.7835 4.6577 5.8687
Panc 10.05 CTRP2 6.1302 7.9294 5.1724 3.5032
Panc 03.27 CTRP2 6.1317 10.1289 4.0744 8.1105
SNU-410 CTRP2 6.1775 10.7307 3.8113 9.1236
Panc 08.13 CTRP2 6.1874 7.6406 5.3621 2.6035
PK-59 CTRP2 6.2197 8.3975 5.0105 4.019
HPAC GDSC1 6.3391 9.2334 3.2737 3.2152
AsPC-1 CTRP2 6.3628 8.1818 5.228 2.8638
BxPC-3 CTRP2 6.3733 8.3856 5.1354 3.2311
PSN1 CTRP2 6.3859 9.2958 4.6938 5.0511
Hs 766T CTRP2 6.4076 8.232 5.2366 2.7556
PSN1 GDSC1 6.4657 11.1684 2.4776 8.1362
HuP-T3 CTRP2 6.4847 7.9983 5.4056 1.9447
CFPAC-1 GDSC1 6.4974 9.29 3.3311 2.6319
SW1990 CTRP2 6.5007 8.4806 5.1824 2.8317
AsPC-1 GDSC1 6.629 12.1231 2.1355 9.9576
SNU-213 CTRP2 6.6625 8.0087 5.5171 1.269
SW1990 GDSC1 6.6638 10.388 2.9466 4.6998
Capan-2 GDSC1 6.6764 8.4373 3.7455 0.5171
Panc 05.04 CTRP2 6.7085 8.5486 5.2931 2.0824
Capan-2 CTRP2 6.7356 8.7475 5.2164 2.3504
Panc 02.03 GDSC1 6.7623 8.0687 3.9049 0.1217
TCC-Pan2 CTRP2 6.8166 9.8349 4.7477 4.1281
KP-3 GDSC1 6.8836 9.4709 3.4407 1.5812
BxPC-3 GDSC1 6.8853 9.2022 3.5456 1.1106
SU.86.86 CTRP2 6.9171 8.7575 5.3278 1.686
HPAF-II CTRP2 6.9711 10.0112 4.77 3.81
YAPC CTRP2 6.9873 11.4625 4.0753 6.6195
Capan-1 CTRP2 6.9978 8.8252 5.3453 1.529
PaTu 8988t CTRP2 7.0323 11.7182 3.9828 6.9272
SUIT-2 CTRP2 7.0761 10.0165 4.8384 3.3895
PK-45H CTRP2 7.3846 9.2515 5.3719 1.0628
PaTu 8902 CTRP2 7.4134 12.4547 3.8961 6.693
L3.3 CTRP2 7.4322 12.0254 4.1165 5.7787
KP-3 CTRP2 7.4516 9.5954 5.2591 1.3794
HuP-T4 CTRP2 7.7445 9.9072 5.2783 1.0729
PaTu 8902 GDSC1 7.7598 16.6779 0.7204 15.157
Panc 02.03 CTRP2 8.6629 10.2309 5.5407 0.1197
CFPAC-1 CTRP2 10.693 28.6968 -1.6804 19.7767
DAN-G CTRP2 11.0659 42.5916 -8.2317 29.8433
Panc 04.03 CTRP2 11.994 24.7498 1.0623 10.8278
⏷ Show the Full List of 67 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 103 Cell Line(s) in Skin Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
SH4 CTRP2 5.3206 10.767 3.0558 13.9809
IGR-1 GDSC1 3.7387 11.6179 0.1772 29.528
A-375 GDSC1 4.1532 8.0942 2.2934 16.3374
COLO 800 GDSC1 4.6014 9.5712 1.9264 17.1866
A101D GDSC1 4.6667 5.8007 3.8465 2.6698
SK-MEL-2 GDSC1 4.6783 8.0216 2.76 11.0086
SK-MEL-1 GDSC1 4.7475 6.2098 3.7048 3.5244
SK-MEL-30 GDSC1 4.777 9.6159 2.044 15.7976
Mel JuSo GDSC1 4.779 6.6497 3.5135 4.8986
COLO 679 GDSC1 5.05 8.8324 2.6409 10.7078
WM1552C GDSC1 5.0679 10.3517 1.9039 15.7519
IGR-37 GDSC1 5.117 6.8146 3.6594 2.9509
WM115 GDSC1 5.1975 6.7449 3.7389 2.2309
DJM-1 GDSC1 5.2134 9.2803 2.5408 10.9407
RPMI-7951 GDSC1 5.2185 10.4539 1.9673 14.8614
SK-MEL-24 GDSC1 5.2345 8.5422 2.9154 8.141
MZ-MEL-2 GDSC1 5.3219 7.4965 3.4704 3.8396
LB373-MEL-D GDSC1 5.345 9.4315 2.5614 10.4074
MZ-MEL-7 GDSC1 5.3696 9.5534 2.5196 10.635
SK-MEL-5 GDSC1 5.4007 7.7427 3.4051 4.1283
MeWo GDSC1 5.4356 7.1785 3.6802 2.1775
A-431 GDSC1 5.4397 12.2205 1.2611 18.4227
SH-4 GDSC1 5.4516 8.5999 3.0353 6.6807
IST-MEL1 GDSC1 5.455 8.386 3.1388 5.9193
WM88 CTRP2 5.4829 9.3253 3.9154 10.0922
G-361 CTRP2 5.4866 7.0267 5.0358 5.4552
HT-144 GDSC1 5.5341 9.5866 2.6185 9.4717
COLO 783 GDSC1 5.546 9.908 2.4715 10.4747
SK-MEL-3 GDSC1 5.5643 7.6682 3.5356 2.8903
451Lu GDSC1 5.5996 8.1417 3.3426 4.135
SK-MEL-28 GDSC1 5.6197 10.2237 2.3701 10.9724
Hs 934.T CTRP2 5.6851 11.1585 3.1821 12.697
CP66-MEL GDSC1 5.6905 7.6071 3.6309 2.0626
Hs 852.T CTRP2 5.7014 8.6054 4.4679 7.3197
UACC-62 GDSC1 5.7268 6.8746 3.9424 0.4293
WM266-4 CTRP2 5.7633 7.7475 4.9485 5.1792
LB2518-MEL GDSC1 5.7779 8.1075 3.4606 2.9904
LOX-IMVI CTRP2 5.7822 8.2467 4.7178 6.1036
G-361 GDSC1 5.7824 7.6379 3.6648 1.7236
RVH-421 GDSC1 5.8171 8.3706 3.366 3.5391
WM115 CTRP2 5.8819 6.5277 5.6568 1.9726
CHL-1 GDSC1 5.9124 10.1359 2.6095 8.5514
M14 GDSC1 5.9255 7.4322 3.8143 0.7896
LOX-IMVI GDSC1 5.933 9.5359 2.904 6.4593
A2058 GDSC1 5.9528 7.2076 3.9099 0.3991
VMRC-MELG GDSC1 6.0125 7.4202 3.8554 0.5525
GAK GDSC1 6.0317 7.4177 3.8641 0.5077
HT-144 CTRP2 6.0581 6.9803 5.5879 1.8926
COLO 792 GDSC1 6.0873 9.165 3.1653 4.3543
Hs 938.T GDSC1 6.1003 7.4769 3.8696 0.4453
MMAc-SF GDSC1 6.1353 7.7076 3.7981 0.6828
A-375 CTRP2 6.163 8.3501 4.9888 4.2134
G-mel GDSC1 6.1732 7.8485 3.7605 0.8057
WT2-iPS GDSC1 6.1824 7.203 3.9957 0.1049
COLO 792 CTRP2 6.1961 7.5082 5.4348 2.2842
IPC-298 GDSC1 6.2311 9.8145 2.9564 5.4604
A-388 GDSC1 6.2553 12.0965 1.9039 12.3176
UACC-257 GDSC1 6.2978 7.4048 3.9677 0.1236
HMV-II GDSC1 6.3404 8.6161 3.5328 1.7232
MeWo CTRP2 6.3464 9.7347 4.4445 6.1637
Mel Ho GDSC1 6.3503 7.7565 3.865 0.3294
Hs 294T CTRP2 6.4106 7.4556 5.6157 1.2057
HMCB CTRP2 6.439 9.1904 4.7869 4.5715
SK-MEL-24 CTRP2 6.5026 7.864 5.4823 1.6109
UACC-257 CTRP2 6.5223 7.9859 5.4373 1.7635
Mel Ho CTRP2 6.5556 9.2195 4.8601 4.0741
SK-MEL-3 CTRP2 6.5587 9.5873 4.6811 4.8109
MDA-MB-435S CTRP2 6.559 7.8834 5.5102 1.4246
IGR-1 CTRP2 6.5619 10.6851 4.14 7.0571
CP50-MEL-B GDSC1 6.5685 7.9658 3.8719 0.2291
Hs 940.T GDSC1 6.5965 8.186 3.8051 0.3816
IGR-39 CTRP2 6.6123 9.0857 4.9671 3.5428
IGR-37 CTRP2 6.6773 10.3933 4.3722 5.8967
COLO 800 CTRP2 6.6788 9.0114 5.0506 3.1002
Hs 936.T CTRP2 6.7004 8.6894 5.2205 2.3827
WM1799 CTRP2 6.7667 8.4299 5.3864 1.643
SK-MEL-5 CTRP2 6.7722 9.9614 4.6544 4.5786
Hs 688(A).T CTRP2 6.7776 9.198 5.0289 3.0436
K029AX CTRP2 6.7845 8.6687 5.2859 2.0108
WM35 GDSC1 6.8654 8.9227 3.6425 0.749
WM793 CTRP2 6.9544 9.2374 5.1276 2.4102
WT2-iPS CTRP2 7.0192 10.0247 4.7963 3.6361
WM278 GDSC1 7.039 9.0382 3.6686 0.56
A2058 CTRP2 7.0673 10.916 4.3994 5.1709
COLO 829 GDSC1 7.0754 8.7024 3.7997 0.222
Hs 895.T CTRP2 7.1352 8.9759 5.3569 1.3426
UACC-62 CTRP2 7.1557 11.8149 4.0247 6.5628
Hs 839.T CTRP2 7.2183 10.7538 4.5816 4.2174
Hs 940.T CTRP2 7.2377 8.8745 5.4565 0.9112
WM793 GDSC1 7.2379 9.0558 3.7363 0.3004
COLO 829 CTRP2 7.2507 14.8297 2.6121 12.052
WM983B CTRP2 7.3286 11.2654 4.4111 4.7453
A101D CTRP2 7.3636 12.4326 3.8717 6.866
SK-MEL-31 CTRP2 7.3951 9.0218 5.4738 0.7377
CJM [Human melanoma] CTRP2 7.5105 8.5004 5.7235 0.1137
SK-MEL-30 CTRP2 7.5112 11.6747 4.3378 4.785
RVH-421 CTRP2 7.5913 17.1591 1.7177 14.7704
SK-MEL-2 CTRP2 7.6363 12.1253 4.2064 5.1354
SK-MEL-1 CTRP2 7.7476 8.9265 5.6614 0.1464
IPC-298 CTRP2 7.8627 14.0731 3.4258 7.9042
Hs 944.T CTRP2 7.9316 11.0577 4.8809 2.2313
Mel JuSo CTRP2 7.9785 14.4972 3.3011 8.2242
SK-MEL-28 CTRP2 10.5852 22.472 1.2365 11.983
⏷ Show the Full List of 103 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 10 Cell Line(s) in Aero Dig Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
OACP4 C GDSC1 4.7986 7.5576 3.0821 8.1634
TE-12 GDSC1 5.2114 9.1599 2.5982 10.533
KYSE-220 GDSC1 5.24 8.8229 2.7831 9.1018
KYSE-50 GDSC1 5.4508 10.4343 2.1478 12.9631
HCE-4 GDSC1 5.7339 10.7107 2.214 11.7135
ESO-26 GDSC1 6.1214 7.9061 3.7158 1.0513
FLO-1 GDSC1 6.1648 10.2309 2.7256 7.1591
OACM5.1 C GDSC1 6.3046 12.5819 1.7047 13.4011
KYAE-1 GDSC1 6.7264 12.8214 1.8701 11.3605
SK-GT-4 GDSC1 7.0346 9.2449 3.5913 0.8203
⏷ Show the Full List of 10 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Ascites Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
COLO 684 GDSC1 5.3558 9.5482 2.5123 10.7265
Cancer Drug Sensitivity Data Curated from 42 Cell Line(s) in Autonomic Ganglia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
IMR-5 GDSC1 -0.7037 11.7747 -4.1217 54.3264
KP-N-YS GDSC1 0.8273 24.2217 -8.6719 48.8274
GOTO GDSC1 2.2315 8.072 0.5101 35.1858
SK-N-MC-IXC GDSC1 3.1807 10.0247 0.4714 30.6863
SJNB-14 GDSC1 3.3762 8.1626 1.566 24.3735
SiMa GDSC1 3.6648 9.695 1.0699 25.8463
KP-N-YN CTRP2 3.6715 9.0793 2.2764 21.0092
SJNB-7 GDSC1 4.2107 8.462 2.1585 17.063
NB1 CTRP2 4.2744 6.9484 3.8079 13.4938
CHP-134 GDSC1 4.4462 13.7311 -0.2795 28.6331
NH-12 GDSC1 4.7436 6.7895 3.4195 5.7263
MHH-NB-11 CTRP2 4.8293 6.325 4.6323 8.7985
SJNB-6 GDSC1 5.1098 7.469 3.3467 5.2587
SJNB-17 GDSC1 5.1822 7.3837 3.4349 4.4226
SK-N-DZ GDSC1 5.2904 6.9052 3.7202 2.1789
MHH-NB-11 GDSC1 5.3258 9.8368 2.3497 11.9562
SK-N-FI GDSC1 5.3299 7.7361 3.364 4.5858
SJNB-12 GDSC1 5.4303 8.3165 3.1556 5.858
TGW GDSC1 5.5819 12.6911 1.1354 18.6725
KP-N-YN GDSC1 5.6055 12.7908 1.1038 18.7702
Kelly GDSC1 5.8011 12.4695 1.4055 16.5323
LA-N-6 GDSC1 5.8451 12.7581 1.296 17.0202
SK-N-BE(2)-M17 GDSC1 5.9053 13.5532 0.9502 18.6904
SK-N-AS GDSC1 5.9461 7.3276 3.8628 0.5723
SK-N-AS CTRP2 6.0338 8.1604 4.9775 4.505
SK-N-SH CTRP2 6.0463 7.0702 5.5331 2.1456
NB(TU)1 GDSC1 6.0642 13.9981 0.8479 18.7561
SK-N-FI CTRP2 6.1494 7.4854 5.4094 2.473
SJNB-13 GDSC1 6.1874 7.8821 3.7538 0.8222
SJNB-10 GDSC1 6.3006 8.1424 3.7022 0.9449
NB1 GDSC1 6.4894 7.8917 3.8689 0.2629
CHP-212 CTRP2 6.5068 7.9032 5.4664 1.6687
SK-N-DZ CTRP2 6.5592 8.0491 5.4318 1.7344
NB69 GDSC1 6.5598 14.6548 0.8808 17.2515
SJNB-5 GDSC1 6.6051 8.3235 3.759 0.5138
CHP-212 GDSC1 6.7005 8.1983 3.8391 0.2562
SK-N-SH GDSC1 6.7239 8.5441 3.7252 0.555
GI-ME-N GDSC1 6.9843 9.2516 3.5683 0.9415
CHP-126 CTRP2 7.1662 8.9555 5.3832 1.22
SK-N-BE(2) CTRP2 7.7459 10.1371 5.1817 1.3784
NH-6 CTRP2 8.0811 9.3816 5.6247 0.1243
KP-N-SI9s CTRP2 8.1842 9.6549 5.5669 0.1787
⏷ Show the Full List of 42 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 8 Cell Line(s) in Biliary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuCC-T1 CTRP2 4.5458 7.8277 3.7242 13.0913
HuCC-T1 GDSC1 5.0225 9.2204 2.4292 12.3242
SNU-478 CTRP2 5.3596 8.5747 4.1714 9.302
SNU-1079 CTRP2 5.7794 7.1836 5.2413 3.9247
HuH-28 CTRP2 6.2264 7.9917 5.218 3.138
SNU-308 CTRP2 6.4467 7.8299 5.4606 1.7776
SNU-1196 CTRP2 6.6201 11.5345 3.7632 8.5196
SNU-869 CTRP2 7.1168 18.9466 0.4637 19.7031
⏷ Show the Full List of 8 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 119 Cell Line(s) in Breast Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MDA-MB-157 CTRP2 1.6448 3.431 1.6376 29.335
HCC1599 GDSC1 3.2489 7.523 1.758 23.7929
MFM-223 GDSC1 3.2637 7.854 1.6116 24.619
HCC2157 GDSC1 3.5695 5.7559 2.9106 14.1841
BT-474 CTRP2 3.6542 8.3416 2.5829 19.8973
CAL-148 GDSC1 3.9543 10.5801 0.8815 25.6088
MRK-nu-1 GDSC1 4.0875 9.1361 1.7168 20.4486
MDA-MB-453 GDSC1 4.1103 7.6139 2.4964 15.0317
DU4475 GDSC1 4.2048 7.0183 2.8749 11.8096
HCC1187 GDSC1 4.5109 8.6243 2.3261 14.776
BT-483 GDSC1 4.6809 6.0927 3.715 3.6328
DU4475 CTRP2 4.6897 6.5529 4.4015 10.0664
MDA-MB-175-VII GDSC1 4.8112 7.1326 3.3006 6.4427
MDA-MB-453 CTRP2 4.8207 7.2068 4.2781 10.1833
HCC202 GDSC1 4.8328 9.501 2.1449 14.9271
UACC-812 GDSC1 5.0253 9.1145 2.4836 11.9261
OCUB-M GDSC1 5.0468 8.744 2.6821 10.4154
CAL-120 GDSC1 5.0783 11.8934 1.1466 20.196
HCC1569 GDSC1 5.1112 8.1878 3.0007 7.8524
MDA-MB-157 GDSC1 5.1209 8.9474 2.6366 10.5245
EFM-19 GDSC1 5.2896 10.5996 1.9485 14.7629
MDA-MB-436 GDSC1 5.2984 10.2718 2.1164 13.6308
CAL-85-1 GDSC1 5.3026 11.8009 1.365 18.2682
MDA-MB-468 GDSC1 5.343 8.4969 3.0119 7.1333
CAL-120 CTRP2 5.3592 9.6227 3.6564 11.4356
Evsa-T GDSC1 5.4942 7.7784 3.4453 3.6433
HCC2218 GDSC1 5.5303 9.3883 2.7113 8.8199
HCC1395 GDSC1 5.5844 9.8705 2.5163 10.0557
BT-474 GDSC1 5.5941 8.2458 3.2915 4.5036
ZR-75-30 GDSC1 5.6818 8.3113 3.3143 4.1582
HCC1500 GDSC1 5.6834 9.6169 2.7051 8.4624
HCC2218 CTRP2 5.7022 9.9085 3.8202 10.0253
CAL-51 GDSC1 5.7096 11.9853 1.5762 15.807
BT-549 GDSC1 5.7354 11.6392 1.7639 14.5989
HCC38 GDSC1 5.8323 10.2358 2.5093 9.4455
MDA-MB-231 GDSC1 5.8599 11.2276 2.0516 12.4332
UACC-893 GDSC1 5.98 8.2254 3.5174 2.3001
ZR-75-30 CTRP2 5.987 7.9092 5.0637 4.2343
COLO 824 GDSC1 5.9913 12.3025 1.6228 14.7299
MCF-7 GDSC1 6.0248 8.3426 3.4907 2.3922
EFM-192A CTRP2 6.0366 7.6381 5.241 3.3919
MDA-MB-361 GDSC1 6.0761 11.0922 2.2634 10.4777
HCC1500 CTRP2 6.0805 9.384 4.4046 6.8227
BT-20 CTRP2 6.0938 7.1097 5.5524 1.9748
HCC1419 GDSC1 6.0985 12.7352 1.4882 15.2215
MDA-MB-468 CTRP2 6.1283 8.6631 4.8043 5.0528
HCC1806 GDSC1 6.1593 13.142 1.3334 15.9307
HCC1954 CTRP2 6.1978 7.844 5.269 2.975
CAL-85-1 CTRP2 6.222 7.7965 5.3116 2.754
EFM-192A GDSC1 6.2304 8.9581 3.3347 3.0162
AU565 CTRP2 6.2339 8.9295 4.7566 5.0582
HCC1428 GDSC1 6.2603 10.7518 2.5431 8.1698
YMB-1-E GDSC1 6.2796 8.7271 3.4577 2.2136
CAL-148 CTRP2 6.3285 8.7091 4.9408 4.1186
JIMT-1 CTRP2 6.3481 9.7785 4.424 6.2468
HCC1937 GDSC1 6.3693 8.5311 3.5804 1.446
HCC1419 CTRP2 6.3917 7.738 5.4667 1.8343
HDQ-P1 GDSC1 6.426 8.4269 3.6466 1.0765
Hs 578T GDSC1 6.4293 9.7673 3.0901 4.2096
SK-BR-3 CTRP2 6.4344 7.9091 5.4137 1.9863
T-47D CTRP2 6.4406 11.4198 3.6793 9.1855
BT-20 GDSC1 6.5292 12.5988 1.8468 11.9772
MDA-MB-361 CTRP2 6.5622 8.2957 5.3156 2.1965
MDA-MB-415 GDSC1 6.5868 13.726 1.3473 14.7262
CAMA-1 GDSC1 6.5932 9.9767 3.0877 3.9416
HCC1395 CTRP2 6.5963 9.8286 4.5903 5.1259
CAL-51 CTRP2 6.612 10.1171 4.4596 5.6424
HCC70 GDSC1 6.6383 12.9135 1.7693 12.1756
HCC1143 CTRP2 6.7156 8.9986 5.0823 2.9173
MDA-MB-415 CTRP2 6.7911 9.3873 4.9469 3.3557
ZR-75-1 CTRP2 6.8095 10.6951 4.3218 5.8895
MDA-MB-231 CTRP2 6.8641 10.0081 4.6971 4.2629
HMC-1-8 CTRP2 6.9498 11.2557 4.1494 6.3749
HCC1937 CTRP2 7.0338 8.9554 5.3074 1.6289
HCC202 CTRP2 7.0883 9.2502 5.2053 1.9485
HCC1428 CTRP2 7.1317 12.4386 3.702 7.9149
KPL-1 CTRP2 7.2541 8.2163 5.7272 0.1786
Hs 578Bst CTRP2 7.2768 10.1764 4.8929 2.9143
HCC1954 GDSC1 7.3271 14.7241 1.3613 12.8743
MDA-MB-330 GDSC1 7.5134 15.5498 1.0927 13.8681
AU565 GDSC1 7.533 10.3584 3.3788 1.2688
CAMA-1 CTRP2 7.5555 13.9167 3.2855 8.921
HDQ-P1 CTRP2 7.6222 9.6262 5.3348 0.9917
HCC1806 CTRP2 8.183 17.1656 2.1496 12.2685
MCF-7 CTRP2 8.6656 10.1362 5.5738 0.0879
T-47D GDSC1 9.0057 19.3332 0.2678 14.6336
BT 440 CTRP2 4.0625 5.8647 3.9278 13.6708
BT 159 CTRP2 5.3961 8.2723 4.3529 8.4687
BT 139 CTRP2 5.5642 7.765 4.7571 6.4151
BT 231 CTRP2 5.6355 11.2074 3.1147 13.0738
BT 145 CTRP2 5.6949 7.449 5.0331 4.9775
BT164 CTRP2 5.9047 7.0685 5.4117 2.9417
BT 228 CTRP2 5.9339 7.97 4.988 4.6584
BT 187 CTRP2 5.9921 7.7379 5.1537 3.8461
BT 239 CTRP2 6.0442 7.3016 5.4157 2.6431
BT 416 CTRP2 6.1262 8.5327 4.8677 4.7902
BT 245 CTRP2 6.1388 9.5246 4.3823 6.8059
BT 482 CTRP2 6.1465 7.4545 5.4226 2.4233
BT 112 CTRP2 6.1943 7.1081 5.6317 1.4657
BT 428 CTRP2 6.2006 8.7646 4.8122 4.8857
BT147 CTRP2 6.353 7.7444 5.4358 2.0203
BT 444 CTRP2 6.3719 8.14 5.2555 2.735
BT 131 CTRP2 6.3878 7.8124 5.4277 1.9999
BT 172 CTRP2 6.3914 7.6802 5.4945 1.7213
BT 359 CTRP2 6.4266 8.613 5.063 3.4435
BT 504 CTRP2 6.5687 9.1549 4.9015 3.8817
BT 179 CTRP2 6.5901 8.2139 5.3738 1.9231
BT 286 CTRP2 6.592 8.6564 5.1618 2.7769
BT 232 CTRP2 6.6316 9.0634 4.9919 3.411
BT 330 CTRP2 6.6333 8.4488 5.2905 2.1963
BT 271 CTRP2 6.6408 10.0811 4.4989 5.4316
BT 422 CTRP2 6.705 9.0402 5.0549 3.0437
BT 224 CTRP2 6.7814 8.799 5.2223 2.265
BT 216 CTRP2 6.7832 8.8152 5.2158 2.2884
BT 320 CTRP2 6.8413 8.309 5.4871 1.1789
BT 333 CTRP2 6.8693 8.5318 5.4024 1.4607
BT 340 CTRP2 7.3994 8.7625 5.5804 0.441
BT 328 CTRP2 7.6046 9.1409 5.5232 0.4751
BT 498 CTRP2 7.7171 8.8642 5.6721 0.1384
⏷ Show the Full List of 119 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Tongue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-38 CTRP2 7.1767 13.0661 3.4267 8.9581
Cancer Drug Sensitivity Data Curated from 99 Cell Line(s) in Central Nervous System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
D283 Med GDSC1 3.6919 7.4493 2.2064 18.8301
SF268 CTRP2 4.2141 7.208 3.6418 14.2984
SF539 CTRP2 4.4139 8.0873 3.4743 14.423
U-251MG GDSC1 4.6093 8.9411 2.2473 14.9851
CAS-1 GDSC1 4.6473 7.6324 2.9294 9.822
YKG-1 GDSC1 4.6728 6.7928 3.3653 6.3629
GB-1 GDSC1 4.8597 9.4355 2.1983 14.4713
PFSK-1 GDSC1 4.9064 8.638 2.6295 11.2394
SF268 GDSC1 5.0267 8.5234 2.7757 9.7837
LN-18 CTRP2 5.0302 6.8326 4.6545 8.1499
8-MG-BA GDSC1 5.0492 10.0023 2.0627 14.7701
D-392MG GDSC1 5.1569 8.3979 2.9309 8.2444
AM-38 GDSC1 5.1623 10.1944 2.0532 14.4735
SNU-466 CTRP2 5.2914 6.5634 5.0397 5.9454
LN-229 GDSC1 5.3412 11.1237 1.7286 15.9934
MOG-G-CCM GDSC1 5.3429 7.9103 3.2905 5.0881
D-542MG GDSC1 5.3783 8.92 2.8326 8.3536
GI-1 GDSC1 5.3816 9.4762 2.5656 10.2728
D-263MG GDSC1 5.4276 11.605 1.5558 16.7724
KNS-60 CTRP2 5.4638 7.0081 5.0218 5.5684
D283 Med CTRP2 5.4837 7.8508 4.6399 7.0831
GB-1 CTRP2 5.5253 9.0684 4.0807 9.3126
SK-MG-1 GDSC1 5.5571 8.8665 2.9782 6.8296
NMC-G1 GDSC1 5.6002 8.1587 3.3352 4.1854
SF539 GDSC1 5.6114 10.806 2.0816 12.9347
SF295 GDSC1 5.6205 10.0204 2.4689 10.2876
YH-13 GDSC1 5.6238 12.1778 1.4191 16.9753
D-247MG GDSC1 5.6703 9.486 2.7587 8.1156
D-336MG GDSC1 5.7152 9.3345 2.86 7.284
SF126 GDSC1 5.7282 10.7924 2.1705 12.0187
TM-31 CTRP2 5.8265 6.3704 5.677 2.0238
GaMG CTRP2 5.8729 8.8874 4.4776 6.9242
Daoy GDSC1 5.9175 10.0657 2.6461 8.2863
ONS-76 GDSC1 5.918 11.4571 1.981 12.7275
KS-1 [Human Krukenberg tumour] GDSC1 5.9229 10.3067 2.5356 9.0341
D-566MG GDSC1 5.93 9.3174 3.0031 5.7795
SW1783 GDSC1 5.9619 10.6708 2.3882 9.9373
42-MG-BA CTRP2 5.9874 27.9684 -4.9652 32.899
T98G CTRP2 5.9901 8.0839 4.9791 4.5838
LNZTA3WT4 GDSC1 6.0399 10.9033 2.3293 10.133
SW1783 CTRP2 6.0559 9.0677 4.5423 6.2912
SNU-201 CTRP2 6.1051 8.3498 4.9419 4.5182
ONS-76 CTRP2 6.1086 8.7015 4.7689 5.2386
MOG-G-UVW GDSC1 6.1181 9.6127 2.9812 5.5264
8-MG-BA CTRP2 6.2148 8.1685 5.1208 3.5658
Onda 11 GDSC1 6.244 11.6064 2.1301 10.9199
M059K CTRP2 6.2662 7.2345 5.6225 1.3884
Hs 683 CTRP2 6.2709 7.284 5.6017 1.4664
SNU-489 CTRP2 6.2715 8.3252 5.0873 3.6056
SNU-738 CTRP2 6.3063 8.8469 4.8549 4.5167
LN-229 CTRP2 6.3197 9.1328 4.7232 5.0444
M059J GDSC1 6.3701 11.539 2.2441 9.8766
LN-405 GDSC1 6.3863 12.1469 1.9672 11.5926
A-172 GDSC1 6.3929 12.6533 1.7301 13.0213
T98G GDSC1 6.4231 10.338 2.8321 5.8947
KALS-1 GDSC1 6.4346 8.6495 3.5631 1.4608
42-MG-BA GDSC1 6.4354 11.0274 2.524 7.8992
LN-18 GDSC1 6.4494 13.1764 1.5177 14.1195
GOS-3 CTRP2 6.5006 8.0905 5.3721 2.0574
GMS-10 CTRP2 6.5131 7.9837 5.4321 1.7974
D-502MG GDSC1 6.5208 8.56 3.6362 1.0373
Daoy CTRP2 6.5468 10.5853 4.1778 6.9257
KNS-81 CTRP2 6.5754 8.2508 5.3462 2.0545
Onda 10 GDSC1 6.5811 11.7592 2.2751 9.1846
A-172 CTRP2 6.6084 10.4015 4.3162 6.2443
GaMG GDSC1 6.6134 13.7083 1.3738 14.5121
DK-MG GDSC1 6.6535 11.945 2.2339 9.2815
CAS-1 CTRP2 6.6717 8.6781 5.2065 2.4793
U-118MG CTRP2 6.6792 9.1927 4.9628 3.4575
SF126 CTRP2 6.6996 11.244 3.9685 7.5331
U-118MG GDSC1 6.7004 8.6924 3.6612 0.7937
SW1088 CTRP2 6.7042 9.0416 5.0537 3.0501
H4 GDSC1 6.7073 15.2804 0.6808 17.8499
CCF-STTG1 CTRP2 6.7202 8.0919 5.514 1.2135
KNS-81-FD GDSC1 6.7253 10.1632 3.0775 3.7873
NMC-G1 CTRP2 6.7257 9.2208 4.982 3.3095
YH-13 CTRP2 6.7291 8.1912 5.4737 1.3547
SNB-75 GDSC1 6.7449 8.7837 3.6453 0.8218
U-251MG CTRP2 6.8149 10.8692 4.2401 6.2178
U-87MG ATCC GDSC1 6.8671 11.9147 2.3785 7.9048
Becker CTRP2 6.8849 10.4816 4.4813 5.1141
SNB-75 CTRP2 6.9065 8.924 5.244 2.0189
KNS-42 CTRP2 6.9293 9.3933 5.0376 2.7977
SNU-626 CTRP2 6.9425 8.4609 5.4771 1.11
DK-MG CTRP2 6.9833 8.5003 5.4825 1.0507
SW1088 GDSC1 7.0488 13.4833 1.7654 11.2347
KINGS-1 GDSC1 7.1248 9.27 3.6179 0.6724
YKG-1 CTRP2 7.1781 10.4886 4.6813 3.8749
KALS-1 CTRP2 7.179 9.1487 5.3047 1.4841
DBTRG-05MG CTRP2 7.2331 9.876 5.0053 2.536
KNS-42 GDSC1 7.2893 15.3518 1.0407 14.6454
D-423MG GDSC1 7.425 9.4088 3.6817 0.3572
U-87MG ATCC CTRP2 7.4338 9.2054 5.4166 0.8823
KG-1-C CTRP2 7.6522 8.9283 5.6239 0.2355
SNU-1105 CTRP2 7.8306 9.1229 5.6227 0.1837
SF295 CTRP2 7.8821 9.1202 5.6431 0.1412
DBTRG-05MG GDSC1 7.9771 15.5082 1.4018 11.2687
Hs 683 GDSC1 8.0204 18.1702 0.1843 17.0017
Becker GDSC1 9.5281 20.742 -0.0616 15.0172
⏷ Show the Full List of 99 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 3 Cell Line(s) in Digestive System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
ETK-1 GDSC1 3.9628 6.9847 2.6806 14.2406
TGBC24TKB GDSC1 6.3975 10.7198 2.6427 7.1995
TGBC1TKB GDSC1 7.5197 16.352 0.7177 15.7088
Cancer Drug Sensitivity Data Curated from 29 Cell Line(s) in Endometrium Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
AN3-CA GDSC1 1.8535 12.0761 -1.765 42.3005
MFE-280 GDSC1 2.5246 9.5364 0.0986 35.1062
JHUEM-2 CTRP2 3.0408 5.9831 2.783 20.9095
MFE-296 GDSC1 3.3534 9.6393 0.8185 28.4126
AN3-CA CTRP2 4.9033 11.1049 2.5099 17.0788
KLE CTRP2 5.4811 7.5124 4.8007 6.4273
HEC-151 CTRP2 5.6552 9.4091 4.0276 9.2575
JHUEM-7 CTRP2 5.6741 6.862 5.2971 3.9375
JHUEM-1 CTRP2 5.7918 6.5407 5.5636 2.5677
HEC-1-A CTRP2 5.8796 7.6819 5.0846 4.364
KLE GDSC1 6.0647 8.8285 3.3018 3.5043
RL95-2 GDSC1 6.1528 7.6773 3.8166 0.5985
MFE-296 CTRP2 6.2688 14.354 2.0751 15.869
MFE-319 GDSC1 6.3565 10.9764 2.4988 8.2432
HEC-6 CTRP2 6.4211 7.6687 5.5207 1.5716
HEC-265 CTRP2 6.4748 9.0002 4.9081 4.0072
EN CTRP2 6.5154 7.7695 5.5357 1.3816
MFE-319 CTRP2 6.5525 10.497 4.2261 6.7149
EN GDSC1 6.5802 12.8935 1.7405 12.4887
HEC-251 CTRP2 6.5977 9.4099 4.7976 4.2648
RL95-2 CTRP2 6.6706 8.297 5.3875 1.7607
HEC-59 CTRP2 6.7662 10.2656 4.5009 5.22
ESS-1 CTRP2 6.8364 8.4847 5.4041 1.4923
EFE-184 CTRP2 6.9624 9.5712 4.9748 3.002
ESS-1 GDSC1 7.8387 18.3366 -0.0156 18.2386
HEC-1-B CTRP2 8.5395 10.355 5.4517 0.2624
HEC-108 CTRP2 10.2514 19.5017 2.4149 8.5009
HEC-50B CTRP2 10.4357 24.8807 -0.0129 15.8976
Ishikawa (Heraklio) 02 ER- CTRP2 14.1958 30.2821 -0.1434 11.8328
⏷ Show the Full List of 29 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 51 Cell Line(s) in Kidney Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
TUHR14TKB CTRP2 3.8064 8.8985 2.4944 19.8283
NCC021 GDSC1 4.7108 7.8213 2.8848 9.9542
KTCTL-13 GDSC1 4.7752 9.3264 2.1867 14.8346
UO-31 CTRP2 4.9401 8.3079 3.8984 11.4042
769-P GDSC1 4.9919 10.6894 1.6779 17.4244
786-O GDSC1 5.0666 10.5476 1.8059 16.3821
KTCTL-140 GDSC1 5.1801 8.8173 2.7431 9.569
TK-10 GDSC1 5.197 11.1095 1.627 17.0679
A-704 GDSC1 5.316 7.5696 3.4329 4.1216
VMRC-RCW GDSC1 5.3529 8.1917 3.1641 5.9884
SW13 GDSC1 5.5209 7.5399 3.5681 2.7563
CAL-54 GDSC1 5.6117 9.8141 2.5622 9.6594
RCC10RGB GDSC1 5.6799 9.2514 2.8762 7.2555
SN12C GDSC1 5.6916 11.3774 1.8603 14.1259
UO-31 GDSC1 5.7285 11.3207 1.9142 13.6803
KTCTL-26A GDSC1 5.7729 13.1558 1.0482 18.567
KTCTL-1M GDSC1 5.8964 11.7897 1.8049 13.8916
LB2241-RCC GDSC1 5.8972 12.674 1.3748 16.4301
HA7-RCC GDSC1 5.9371 14.9818 0.2709 21.8042
BFTC-909 GDSC1 5.9919 8.316 3.485 2.4773
ACHN GDSC1 6.0008 14.3134 0.6469 19.9141
VMRC-RCZ GDSC1 6.0031 9.0687 3.16 4.5548
A-498 GDSC1 6.0174 7.2583 3.9166 0.3423
SW156 GDSC1 6.0175 8.8548 3.2639 3.8361
TUHR4TKB CTRP2 6.0942 8.9434 4.6362 5.8238
LB1047-RCC GDSC1 6.1024 14.4141 0.6718 19.5098
KTCTL-195 GDSC1 6.1133 8.0101 3.671 1.2763
RXF 393L GDSC1 6.1649 9.0298 3.2685 3.5407
BB65-RCC GDSC1 6.2074 13.0622 1.4059 15.3939
LB996-RCC GDSC1 6.2993 9.4195 3.1713 3.9236
CAL-54 CTRP2 6.3446 7.8552 5.3753 2.2833
786-O CTRP2 6.4558 9.0622 4.8631 4.2259
SNU-1272 CTRP2 6.4737 7.7295 5.5272 1.4716
VMRC-RCZ CTRP2 6.5346 10.6954 4.1137 7.2136
KMRC-1 GDSC1 6.59 13.9713 1.2316 15.349
Caki-2 CTRP2 6.6518 7.9538 5.5358 1.2105
KMRC-2 CTRP2 6.6729 9.8666 4.6284 4.8432
KTCTL-21 GDSC1 6.6839 16.414 0.1134 20.461
KMRC-1 CTRP2 6.7051 9.7142 4.7267 4.3863
OS-RC-2 CTRP2 6.9083 9.8422 4.8084 3.7457
BFTC-909 CTRP2 6.9861 9.8537 4.8559 3.4439
OS-RC-2 GDSC1 7.014 14.54 1.2447 14.2287
KMRC-20 GDSC1 7.2219 14.7881 1.2634 13.64
ACHN CTRP2 7.3362 11.1845 4.4549 4.5597
VMRC-RCW CTRP2 7.4015 8.8694 5.5389 0.5485
TUHR10TKB CTRP2 7.4895 8.5717 5.6901 0.17
RCC10RGB CTRP2 7.5695 9.0183 5.5555 0.4146
KMRC-20 CTRP2 7.6258 13.4979 3.5392 7.8056
769-P CTRP2 8.4128 17.1818 2.3047 11.3544
Caki-1 CTRP2 8.4974 12.5424 4.5402 2.8708
Caki-1 GDSC1 9.2805 22.3188 -0.9556 18.8017
⏷ Show the Full List of 51 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 87 Cell Line(s) in Large Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H716 CTRP2 1.6349 3.1667 1.6324 29.3853
NCI-H716 GDSC1 3.3647 9.2391 1.0262 27.364
HCT 116 GDSC1 4.4176 7.1035 3.01 9.9853
HCT 15 CTRP2 4.4835 7.2929 3.8906 12.6008
LoVo GDSC1 4.8014 7.4595 3.1326 7.7662
HT115 GDSC1 5.0491 6.5844 3.7239 2.642
LS513 GDSC1 5.1103 6.9796 3.5786 3.5467
SW1417 GDSC1 5.1225 7.0788 3.5399 3.7985
COLO205 GDSC1 5.1353 8.5903 2.8218 9.1183
CCK-81 GDSC1 5.2021 9.4053 2.4712 11.4718
RKO GDSC1 5.2178 7.3843 3.4575 4.1726
SW948 GDSC1 5.2245 7.3275 3.4882 3.934
HT115 CTRP2 5.2658 6.488 5.0427 6.0042
LS123 GDSC1 5.39 8.8651 2.8671 8.0701
LS411N GDSC1 5.3983 7.6871 3.4293 3.9616
SW1116 GDSC1 5.4005 7.3464 3.5859 2.8689
SNU-C1 CTRP2 5.4059 8.806 4.101 9.49
RCM-1 [Human ESC] GDSC1 5.4659 12.613 1.0869 19.284
CW-2 GDSC1 5.4784 10.907 1.9364 14.2676
HCT 15 GDSC1 5.5291 9.2781 2.7633 8.4502
LoVo CTRP2 5.5605 8.3132 4.4852 7.5519
T84 CTRP2 5.5745 7.741 4.7785 6.3035
NCI-H747 CTRP2 5.5798 12.097 2.6227 15.1593
SNU-175 GDSC1 5.6576 10.5096 2.2582 11.6287
COLO 320 CTRP2 5.6591 8.0311 4.7141 6.3827
SW48 GDSC1 5.6763 8.4347 3.2546 4.5839
COLO 320HSR GDSC1 5.6764 11.2327 1.92 13.7926
SNU-C1 GDSC1 5.7667 10.6115 2.2846 11.1504
MDST8 GDSC1 5.7751 8.3255 3.3623 3.6445
GP5d GDSC1 5.778 8.1135 3.458 3.0068
HT-29 GDSC1 5.7863 10.0754 2.555 9.2481
HT-55 GDSC1 5.8234 9.9174 2.6547 8.46
LS180 CTRP2 5.9249 8.8268 4.5524 6.5058
HCC2998 GDSC1 5.9446 9.1635 3.0825 5.2015
SW1463 GDSC1 5.9446 8.3851 3.4301 2.8949
LS1034 GDSC1 5.9573 9.7833 2.8041 7.0968
COLO205 CTRP2 6.0327 12.0079 3.0529 12.5242
LS180 GDSC1 6.0327 9.6463 2.9144 6.165
NCI-H747 GDSC1 6.0401 8.4937 3.4341 2.7121
SW626 GDSC1 6.0633 9.7999 2.8623 6.4544
KM12 GDSC1 6.1342 10.9343 2.3766 9.582
OUMS-23 CTRP2 6.1529 9.4867 4.4128 6.651
C2BBe1 CTRP2 6.1574 7.6325 5.3424 2.7395
C2BBe1 GDSC1 6.1946 11.046 2.3632 9.5231
SW620 CTRP2 6.2019 8.0243 5.1825 3.33
CaR-1 GDSC1 6.287 12.1078 1.9198 12.1377
SNU-C5 CTRP2 6.2929 8.7862 4.8747 4.4575
SW1417 CTRP2 6.3048 7.6767 5.4338 2.1055
SNU-61 CTRP2 6.3147 8.6485 4.9602 4.0618
SNU-407 CTRP2 6.3475 8.133 5.2407 2.8364
SNU-C4 CTRP2 6.3838 7.5842 5.5357 1.5651
SW620 GDSC1 6.4067 10.9874 2.5248 7.9579
T84 GDSC1 6.4191 8.6802 3.5437 1.5749
SW948 CTRP2 6.4282 7.9772 5.3762 2.1489
HCT 8 CTRP2 6.4375 9.0517 4.8545 4.2921
SNU-C5 GDSC1 6.4487 10.1181 2.9456 5.1024
HT-55 CTRP2 6.4529 9.4414 4.6731 5.0219
SW48 CTRP2 6.4561 9.1425 4.8236 4.3895
SNU-81 GDSC1 6.4721 8.0709 3.7989 0.4617
SNU-1040 GDSC1 6.4814 7.8466 3.8817 0.2368
DLD-1 CTRP2 6.488 8.1071 5.3553 2.1443
SNU-61 GDSC1 6.5125 8.2276 3.7576 0.5724
SK-CO-1 CTRP2 6.5214 8.2788 5.2954 2.3381
RKO CTRP2 6.5218 9.0181 4.9342 3.822
SNU-407 GDSC1 6.5316 11.3033 2.4558 8.1315
NCI-H508 CTRP2 6.5858 11.7017 3.6533 9.0336
LS513 CTRP2 6.6068 10.8178 4.1086 7.1101
CL-11 GDSC1 6.6174 8.9302 3.5345 1.4074
GP2d CTRP2 6.65 8.303 5.3711 1.8524
LS1034 CTRP2 6.6659 9.7248 4.6929 4.5878
SNU-C2B GDSC1 6.7809 10.7949 2.8322 5.2081
CL-11 CTRP2 6.8371 8.8058 5.2552 2.0629
RCM-1 [Human ESC] CTRP2 6.8633 8.7829 5.2826 1.9236
LS123 CTRP2 6.8639 8.8227 5.2644 1.9933
HCC-56 CTRP2 6.8848 13.642 2.9212 11.4747
MDST8 CTRP2 6.948 9.3994 5.047 2.7356
HT-29 CTRP2 6.9931 15.8457 1.9102 15.1243
COLO 678 GDSC1 7.003 8.5601 3.8227 0.1993
COLO201 CTRP2 7.0924 13.7862 3.0085 10.7717
LS411N CTRP2 7.2856 11.12 4.4517 4.6431
SW837 GDSC1 7.4247 8.9505 3.8366 0.099
SNU-503 CTRP2 7.6056 9.391 5.4237 0.7397
COLO 678 CTRP2 7.7133 9.5714 5.4014 0.7332
SNU-C2A CTRP2 8.3306 10.5599 5.2892 0.6753
CW-2 CTRP2 8.5551 10.5765 5.3772 0.3876
KM12 CTRP2 9.6215 22.1978 0.7196 14.8935
HCT 116 CTRP2 10.2429 21.8445 1.3097 12.1936
⏷ Show the Full List of 87 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Leukemia Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MO-T GDSC1 4.4405 8.1387 2.5114 13.6865
Cancer Drug Sensitivity Data Curated from 36 Cell Line(s) in Liver Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Hep 3B2.1-7 GDSC1 3.7991 7.8141 2.123 18.9546
Huh-7 GDSC1 4.1536 8.9248 1.8787 19.1601
SNU-475 GDSC1 4.6939 7.7446 2.9098 9.8185
JHH-2 GDSC1 4.7593 7.1646 3.2466 7.0165
SNU-423 GDSC1 4.9602 6.5302 3.6936 3.0648
JHH-1 GDSC1 4.9941 6.2275 3.8539 1.8515
JHH-6 GDSC1 5.0734 9.0831 2.5349 11.4076
Li-7 CTRP2 5.145 9.5281 3.506 12.5313
SNU-398 GDSC1 5.2038 8.9009 2.7193 9.6746
Hep-G2/C3A GDSC1 5.466 7.8084 3.4147 3.9165
JHH-5 CTRP2 5.4817 7.8475 4.6397 7.0885
HLF CTRP2 5.5079 6.568 5.264 4.4882
JHH-7 GDSC1 5.6492 9.2082 2.8767 7.3287
PLC/PRF/5 CTRP2 5.7128 6.9901 5.2731 3.9442
SK-HEP-1 GDSC1 5.7463 8.4345 3.2964 4.1482
HuH-6 CTRP2 5.8362 10.2415 3.7699 9.9616
JHH-1 CTRP2 5.8936 6.7789 5.545 2.4096
JHH-4 CTRP2 6.0414 11.072 3.5281 10.5609
SNU-761 CTRP2 6.158 7.6668 5.3258 2.8082
HLE GDSC1 6.1633 10.5684 2.5674 8.2327
HuH-1 CTRP2 6.2117 8.1269 5.1391 3.4944
SNU-878 CTRP2 6.3593 9.133 4.7541 4.8454
HuH-1 GDSC1 6.5599 7.9126 3.8871 0.2004
JHH-2 CTRP2 6.5611 9.512 4.7201 4.6454
SNU-449 GDSC1 6.5651 12.882 1.736 12.5529
SNU-423 CTRP2 6.6061 8.2066 5.388 1.8448
SK-HEP-1 CTRP2 6.747 8.9364 5.1337 2.6654
SNU-182 CTRP2 6.9037 9.2282 5.0991 2.5888
SNU-449 CTRP2 6.9504 9.3511 5.0714 2.6359
JHH-6 CTRP2 7.0271 8.0572 5.6915 0.3621
SNU-387 GDSC1 7.2185 8.9218 3.7754 0.2283
Hep 3B2.1-7 CTRP2 7.4799 13.4698 3.4494 8.3859
SNU-398 CTRP2 8.0496 10.2406 5.2886 0.8346
SNU-387 CTRP2 8.2284 10.0998 5.4219 0.4208
JHH-4 GDSC1 8.2324 35.1363 -7.96 34.5124
Hep-G2 CTRP2 8.2938 26.0392 -2.1458 24.3207
⏷ Show the Full List of 36 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 306 Cell Line(s) in Lung Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NCI-H1581 GDSC1 1.7388 5.9113 0.9522 36.379
IST-SL2 GDSC1 2.8889 8.0931 1.1405 29.0174
NCI-H2795 GDSC1 3.5025 6.4477 2.5174 17.4276
NCI-H1581 CTRP2 3.8947 8.9992 2.5384 19.4287
SBC-3 GDSC1 4.4393 7.5343 2.8124 11.4315
UMC-11 GDSC1 4.4483 8.0591 2.5576 13.3182
NCI-H810 CTRP2 4.471 6.8594 4.052 12.0116
NCI-H2810 GDSC1 4.509 7.2942 2.9886 9.8324
NCI-H1694 CTRP2 4.5155 8.8512 3.2266 15.1538
NCI-H1341 CTRP2 4.5554 6.804 4.1633 11.3504
HOP-62 GDSC1 4.5689 7.4338 2.9668 9.797
NCI-H2803 GDSC1 4.5935 8.9842 2.2131 15.2793
NCI-H1155 GDSC1 4.5938 8.8165 2.297 14.6898
NCI-H1155 CTRP2 4.6838 7.9719 3.7994 12.4384
NCI-H2081 CTRP2 4.7382 7.0751 4.2479 10.522
ABC-1 GDSC1 4.7984 7.8354 2.9447 9.2161
NCI-H510A GDSC1 4.8218 8.0783 2.8424 9.9191
IA-LM GDSC1 4.8418 7.9737 2.9091 9.3501
NCI-H1703 CTRP2 4.8441 7.7043 4.0823 10.8998
BEN GDSC1 4.9078 8.7561 2.5722 11.656
NCI-H226 GDSC1 4.9079 7.258 3.309 6.0957
NCI-H520 GDSC1 4.9161 7.285 3.3016 6.1283
NCI-H526 CTRP2 4.9495 7.4261 4.3141 9.7052
NCI-H1770 GDSC1 4.9841 8.703 2.6558 10.8022
Ms-1 GDSC1 4.994 11.0025 1.5238 18.3461
PC-14 GDSC1 5.005 8.5704 2.7366 10.1405
A-427 GDSC1 5.0163 10.6131 1.7346 16.9937
NCI-H187 GDSC1 5.0511 7.8054 3.1441 6.9426
HCC78 GDSC1 5.088 8.3261 2.9168 8.5481
SBC-5 GDSC1 5.0987 6.3249 3.8697 1.5489
NCI-H211 CTRP2 5.1031 7.3655 4.4969 8.5834
LK-2 GDSC1 5.1167 10.0691 2.0808 14.434
DMS 53 GDSC1 5.1249 9.6446 2.2965 12.9375
NCI-H1781 GDSC1 5.1279 7.7839 3.2078 6.2506
COR-L321 GDSC1 5.1301 9.0104 2.6123 10.6736
NCI-H2171 GDSC1 5.1598 8.1388 3.0586 7.2819
NCI-H2444 GDSC1 5.1801 7.6646 3.3003 5.4219
DV-90 CTRP2 5.2127 7.1658 4.6978 7.5012
DMS 53 CTRP2 5.2359 8.0558 4.3051 9.037
NCI-H290 GDSC1 5.2388 9.5632 2.4206 11.7199
NCI-H526 GDSC1 5.2457 9.0828 2.6606 9.9807
NCI-H1975 GDSC1 5.2684 8.9846 2.7246 9.4492
NCI-H1694 GDSC1 5.2697 9.8699 2.2928 12.5187
COR-L311 GDSC1 5.2895 10.1174 2.1856 13.1916
NCI-H2818 GDSC1 5.292 9.7015 2.3915 11.7651
NCI-H1436 GDSC1 5.2998 10.2625 2.1219 13.589
NCI-H2087 CTRP2 5.3089 6.4554 5.1014 5.6594
LB647-SCLC GDSC1 5.3091 7.3453 3.5322 3.4297
COR-L303 GDSC1 5.3177 8.8734 2.8132 8.6624
NCI-H3122 GDSC1 5.3215 11.2212 1.6658 16.4396
SBC-1 GDSC1 5.3239 10.7635 1.8932 15.0126
NCI-H2081 GDSC1 5.3245 11.6845 1.4392 17.7746
NCI-H1666 CTRP2 5.3478 6.654 5.0612 5.7093
NCI-H1666 GDSC1 5.3494 7.6034 3.4379 4.0098
COR-L88 GDSC1 5.3509 9.687 2.441 11.2441
NCI-H2106 CTRP2 5.3664 7.842 4.5328 7.7961
CAL-12T GDSC1 5.3692 8.7217 2.9218 7.7254
NCI-H211 GDSC1 5.3933 9.3406 2.6396 9.7099
DMS 454 CTRP2 5.4087 8.1872 4.4061 8.2203
NCI-H1304 GDSC1 5.4154 9.9373 2.3651 11.5865
VMRC-LCD CTRP2 5.4181 9.4436 3.7983 10.719
NCI-H2135 GDSC1 5.4221 8.9718 2.8377 8.198
NCI-H524 GDSC1 5.425 8.4087 3.1085 6.2142
NCI-H2029 GDSC1 5.432 8.2015 3.2109 5.4519
NCI-H1915 CTRP2 5.436 6.7986 5.0891 5.3683
NCI-H2066 GDSC1 5.4379 11.1577 1.7836 15.3555
IST-SL1 GDSC1 5.4476 9.4424 2.6283 9.6398
Calu-6 CTRP2 5.4977 10.3845 3.4034 12.181
LC-2/ad GDSC1 5.5146 11.2386 1.8002 15.0217
NCI-H841 CTRP2 5.5224 7.937 4.6343 7.0183
EMC-BAC-1 GDSC1 5.5411 9.0709 2.8705 7.6468
Lu-99 CTRP2 5.5467 8.6966 4.2837 8.4207
NCI-H1573 CTRP2 5.5581 6.6286 5.289 4.2583
CPC-N GDSC1 5.5727 10.1667 2.3649 11.1389
COR-L95 GDSC1 5.5757 7.5057 3.6136 2.3608
NCI-H209 GDSC1 5.5883 10.7252 2.1045 12.8508
NCI-H446 CTRP2 5.5906 7.1131 5.097 4.9543
NCI-H69 CTRP2 5.5925 8.2342 4.5533 7.198
NCI-H1703 GDSC1 5.5954 12.6539 1.1638 18.4795
EKVX GDSC1 5.6021 9.1958 2.8515 7.6274
HCC15 CTRP2 5.623 10.0884 3.6613 10.8508
LCLC-97TM1 GDSC1 5.6479 11.3564 1.8392 14.3848
HCC44 CTRP2 5.6534 9.2918 4.0844 9.0242
NCI-H2141 GDSC1 5.6606 8.4491 3.2385 4.7303
LCLC-103H GDSC1 5.6681 8.6764 3.1381 5.4204
DMS 79 CTRP2 5.6824 9.6636 3.9249 9.6297
NCI-H345 GDSC1 5.6834 6.8269 3.9425 0.4588
NCI-H146 GDSC1 5.694 9.3583 2.8349 7.5143
NCI-H847 GDSC1 5.6964 11.1362 1.9813 13.3434
EPLC-272H GDSC1 5.6981 10.0997 2.4839 9.9739
NCI-H2196 CTRP2 5.6983 6.6255 5.4318 3.3314
NCI-H460 GDSC1 5.6999 8.9116 3.0486 5.9815
NCI-H1573 GDSC1 5.704 8.0481 3.4455 3.2253
NCI-H2869 GDSC1 5.7139 10.2183 2.4377 10.2503
NCI-H82 GDSC1 5.7151 10.7978 2.1587 12.1327
NCI-H2291 GDSC1 5.7173 8.5477 3.2276 4.6837
NCI-H64 GDSC1 5.7245 11.9564 1.6011 15.6162
HOP-92 CTRP2 5.7392 7.9961 4.8038 5.8353
NCI-H1092 GDSC1 5.7408 10.4604 2.3396 10.8486
Lu-65 GDSC1 5.741 9.5117 2.793 7.6952
Lu-135 GDSC1 5.7836 10.8592 2.1767 11.8247
NCI-H358 GDSC1 5.7908 9.844 2.6681 8.4485
NCI-H1693 CTRP2 5.7962 7.2855 5.2065 4.032
NCI-H441 GDSC1 5.8048 10.3357 2.443 9.9724
NCI-H2170 CTRP2 5.8089 7.4641 5.1298 4.3245
COR-L23 GDSC1 5.815 10.9991 2.1308 12.0407
NCI-H841 GDSC1 5.8268 8.8448 3.1575 4.9356
HOP-62 CTRP2 5.8278 7.1975 5.2787 3.6627
EBC-1 CTRP2 5.8411 7.8546 4.9648 4.9462
RERF-LC-A1 CTRP2 5.8418 8.9309 4.4291 7.191
NCI-H838 GDSC1 5.8473 9.2983 2.9609 6.2587
NCI-H810 GDSC1 5.8619 10.209 2.5417 9.1462
NCI-H1793 CTRP2 5.8769 6.8259 5.5066 2.6063
NCI-H1734 GDSC1 5.8774 12.8477 1.2756 17.0406
NCI-H196 GDSC1 5.8872 8.8918 3.1721 4.7081
RERF-LC-MS CTRP2 5.8911 7.5045 5.1829 3.9283
EBC-1 GDSC1 5.8975 10.8553 2.2567 10.986
NCI-H1568 CTRP2 5.9056 6.8107 5.5402 2.4035
SBC-5 CTRP2 5.9093 6.6342 5.6305 2.0194
NCI-H292 GDSC1 5.9112 8.8986 3.1832 4.5838
NCI-H2029 CTRP2 5.9127 6.7751 5.5642 2.2878
Lu-165 GDSC1 5.9147 9.7994 2.7695 7.4371
NCI-H2023 CTRP2 5.9186 8.7521 4.5843 6.3842
NCI-H661 CTRP2 5.9281 9.6181 4.1597 8.1479
NCI-H1092 CTRP2 5.9349 6.9565 5.4941 2.5334
NCI-H2373 GDSC1 5.9355 10.9057 2.2583 10.8755
COLO 668 CTRP2 5.9384 7.8958 5.0289 4.4776
NCI-H3255 GDSC1 5.9747 9.2433 3.0641 5.2637
NCI-H661 GDSC1 5.9771 9.2957 3.0416 5.4129
A-549 GDSC1 5.9793 9.0492 3.155 4.6366
NCI-H1105 CTRP2 5.985 7.8463 5.0935 4.1131
NCI-H69 GDSC1 5.9934 10.5647 2.4595 9.3757
Lu-65 CTRP2 5.9952 7.92 5.0653 4.2112
NCI-H2722 GDSC1 5.9955 11.0452 2.232 10.8925
NCI-H2009 GDSC1 6.002 10.7983 2.3541 10.0637
NCI-H2087 GDSC1 6.008 8.8081 3.2793 3.7532
ChaGo-K-1 CTRP2 6.0255 7.1688 5.4664 2.4663
NCI-H2347 GDSC1 6.0275 8.8856 3.2559 3.8705
NCI-H1650 GDSC1 6.0407 9.0238 3.2018 4.2021
SHP-77 CTRP2 6.0464 7.0814 5.5276 2.1683
NCI-H1341 GDSC1 6.0464 8.0326 3.6307 1.5633
HCC1588 CTRP2 6.0506 9.4044 4.3696 7.0274
HCC2935 CTRP2 6.057 8.0841 5.035 4.2185
Calu-3 CTRP2 6.0652 7.9599 5.1039 3.9131
NCI-H23 CTRP2 6.0658 7.3269 5.4209 2.5799
HCC827 CTRP2 6.0843 7.4349 5.3821 2.7078
NCI-H1836 GDSC1 6.0912 12.1616 1.7607 13.629
NCI-H1437 GDSC1 6.1025 9.1082 3.1992 4.1018
NCI-H23 GDSC1 6.1028 10.062 2.7654 7.0281
SHP-77 GDSC1 6.1099 7.6807 3.7977 0.7042
SW1573 GDSC1 6.1118 11.371 2.1543 11.0994
NCI-H446 GDSC1 6.1297 10.4724 2.591 8.1522
COLO 668 GDSC1 6.1383 8.8104 3.3496 3.0747
NCI-H1915 GDSC1 6.1391 9.7572 2.9279 5.8429
NCI-H2196 GDSC1 6.1436 13.7556 1.0237 17.6397
ChaGo-K-1 GDSC1 6.1458 10.8141 2.4409 9.1245
NCI-H1651 GDSC1 6.1474 9.1403 3.2102 3.947
EMC-BAC-2 GDSC1 6.1474 11.4739 2.129 11.1724
NCI-H838 CTRP2 6.1513 8.0945 5.107 3.7389
HCC827 GDSC1 6.1532 11.2354 2.2464 10.3942
DMS 114 GDSC1 6.1661 12.6116 1.5952 14.4158
NCI-H1048 GDSC1 6.1749 11.5434 2.1142 11.1971
COR-L51 CTRP2 6.1853 7.9185 5.222 3.1944
NCI-H2342 GDSC1 6.1961 9.9748 2.8626 6.1628
NCI-H2170 GDSC1 6.2097 11.0871 2.3535 9.55
Lu-139 GDSC1 6.2102 8.443 3.5413 1.8402
NCI-H2122 GDSC1 6.2203 9.8332 2.9415 5.5821
LXF 289 CTRP2 6.2219 8.047 5.1869 3.2759
NCI-H522 GDSC1 6.228 10.9161 2.4457 8.8946
DMS 273 CTRP2 6.2384 7.4374 5.5023 1.9307
NCI-H2595 GDSC1 6.2425 8.3904 3.5781 1.6025
NCI-H1184 CTRP2 6.2447 8.4565 5.001 4.0141
HCC2279 CTRP2 6.2461 8.1114 5.1738 3.2882
SK-MES-1 GDSC1 6.2489 8.2548 3.6355 1.3047
HCC95 CTRP2 6.2522 8.998 4.737 5.1075
COR-L95 CTRP2 6.3198 8.3057 5.1342 3.3262
NCI-H2228 GDSC1 6.3231 10.4446 2.7239 6.8208
NCI-H650 CTRP2 6.3236 8.299 5.1405 3.2933
NCI-H2804 GDSC1 6.3293 12.2704 1.8705 12.3335
NCI-H2405 GDSC1 6.3319 9.4153 3.191 3.7419
NCI-H2461 GDSC1 6.3376 11.2107 2.3775 9.0858
Lu-134-A GDSC1 6.3386 9.7257 3.058 4.581
NCI-H727 CTRP2 6.34 8.6591 4.9745 3.9582
HCC15 GDSC1 6.3421 10.9699 2.4928 8.3161
NCI-H650 GDSC1 6.3444 11.9822 2.0178 11.3809
NCI-H1435 CTRP2 6.3878 7.6086 5.5267 1.5957
NCI-H2110 CTRP2 6.3955 8.6048 5.0437 3.5754
MOR/CPR CTRP2 6.396 14.8029 1.9546 16.0685
LK2 CTRP2 6.4271 10.447 4.1534 7.2373
NCI-H2731 GDSC1 6.4452 12.0975 2.0293 11.0598
NCI-H2591 GDSC1 6.4566 13.7005 1.2704 15.4837
NCI-H1838 GDSC1 6.4567 13.4045 1.4131 14.6941
NCI-H647 GDSC1 6.4581 10.4765 2.7899 6.1007
HCC44 GDSC1 6.4635 11.7719 2.1947 9.9712
NCI-H1869 CTRP2 6.483 8.0045 5.4014 1.9641
NCI-H522 CTRP2 6.4947 8.0969 5.3649 2.0952
PC-14 CTRP2 6.5027 8.8687 4.9936 3.6071
NCI-H2369 GDSC1 6.5112 12.9616 1.6622 13.1237
RERF-LC-Ad2 CTRP2 6.5179 7.7049 5.5678 1.2525
NCI-H2342 CTRP2 6.524 8.3803 5.248 2.5274
KNS-62 CTRP2 6.5521 8.0221 5.4399 1.7117
NCI-H2126 CTRP2 6.5613 9.2513 4.8487 4.112
NCI-H1993 GDSC1 6.572 13.0311 1.6696 12.9275
NCI-H1355 GDSC1 6.5774 12.9486 1.7125 12.6615
NCI-H1755 GDSC1 6.578 8.7947 3.5701 1.2799
Calu-3 GDSC1 6.5868 8.7452 3.5932 1.1666
Sq-1 CTRP2 6.6017 8.0508 5.459 1.57
Calu-6 GDSC1 6.6077 13.327 1.5523 13.519
NCI-H2172 GDSC1 6.6204 8.4103 3.7334 0.5887
NCI-H2110 GDSC1 6.6279 10.6886 2.793 5.7438
NCI-H1563 GDSC1 6.6349 13.4727 1.501 13.744
LOU-NH91 GDSC1 6.6394 13.9005 1.2993 14.8561
CAL-12T CTRP2 6.6417 18.7521 0.1812 21.4143
NCI-H1435 GDSC1 6.6459 14.1178 1.1993 15.38
PaCa-3 GDSC1 6.6567 12.3771 2.0341 10.5238
NCI-H1876 GDSC1 6.658 8.3863 3.7568 0.492
NCI-H520 CTRP2 6.6585 9.73 4.685 4.6323
COLO 699 CTRP2 6.6587 9.2109 4.9393 3.5849
SW1271 CTRP2 6.6762 9.0376 5.0361 3.163
NCI-H1568 GDSC1 6.6833 9.2842 3.4235 1.8849
NCI-H513 GDSC1 6.6957 9.1484 3.4836 1.5706
SW1271 GDSC1 6.7005 8.8303 3.6093 0.9989
NCI-H2030 GDSC1 6.7043 11.394 2.5188 7.3539
NCI-H2405 CTRP2 6.7412 9.3048 4.9521 3.408
NCI-H1651 CTRP2 6.7535 8.4918 5.3491 1.804
NCI-H1299 GDSC1 6.76 11.8927 2.3239 8.4766
NCI-H647 CTRP2 6.8059 8.4073 5.4211 1.4636
NCI-H1355 CTRP2 6.8225 9.6969 4.8189 3.8289
DMS 114 CTRP2 6.8245 10.0251 4.6608 4.4716
NCI-H596 GDSC1 6.8348 16.1512 0.3481 19.0609
BEN CTRP2 6.8761 20.5952 -0.5501 22.9886
DMS 273 GDSC1 6.8874 8.3056 3.8685 0.1502
NCI-H720 GDSC1 6.8971 17.7505 -0.3859 21.9153
NCI-H889 CTRP2 6.9116 11.1139 4.191 6.2647
COR-L105 CTRP2 6.9143 8.6873 5.3583 1.5745
NCI-H2023 GDSC1 6.9173 13.9069 1.4815 13.1642
NCI-H226 CTRP2 6.9412 10.3139 4.603 4.5307
NCI-H322 CTRP2 6.9555 9.1231 5.1819 2.1979
HARA [Human squamous cell lung carcinoma] CTRP2 6.9584 10.7113 4.4219 5.2442
NCI-H1650 CTRP2 6.9728 9.1098 5.199 2.1103
NCI-H727 GDSC1 6.9769 8.5222 3.8264 0.1993
HARA [Human squamous cell lung carcinoma] GDSC1 6.9813 12.414 2.2188 8.6588
NCI-H1734 CTRP2 6.9823 8.6801 5.4018 1.339
SK-LU-1 GDSC1 6.9905 14.2629 1.3607 13.658
NCI-H196 CTRP2 6.9991 9.8608 4.8613 3.404
NCI-H358 CTRP2 7.0114 10.5214 4.5516 4.6353
RERF-LC-KJ GDSC1 7.0192 12.4532 2.2236 8.5492
LOU-NH91 CTRP2 7.0608 8.8273 5.3809 1.3325
NCI-H1563 CTRP2 7.0745 8.8735 5.3681 1.3643
RERF-LC-Ad1 CTRP2 7.0855 7.9158 5.7706 0.1552
NCI-H1792 CTRP2 7.1335 9.1789 5.2649 1.6764
NCI-H1299 CTRP2 7.141 10.3756 4.7104 3.8101
Calu-1 CTRP2 7.1462 10.1921 4.8012 3.4421
HCC1438 CTRP2 7.1633 11.443 4.2111 5.7924
LCLC-103H CTRP2 7.1755 10.8602 4.5015 4.5989
LC-1/sq-SF CTRP2 7.1797 9.5425 5.1265 2.139
LUDLU-1 CTRP2 7.1973 8.768 5.481 0.8656
HCC366 CTRP2 7.2115 9.4441 5.1906 1.8643
NCI-H1688 GDSC1 7.214 15.9475 0.7069 16.4736
NCI-H322M GDSC1 7.2372 9.426 3.6051 0.6498
NCI-H1944 GDSC1 7.2622 14.8232 1.2729 13.4962
A-549 CTRP2 7.2697 10.0007 4.9702 2.6257
KNS-62 GDSC1 7.3093 12.6432 2.3083 7.4503
EKVX CTRP2 7.3111 12.6648 3.7213 7.5541
HCC33 GDSC1 7.3145 18.4327 -0.4219 21.0421
HCC1833 CTRP2 7.3189 10.4494 4.7919 3.2531
NCI-H1648 GDSC1 7.3284 9.1785 3.7265 0.2921
NCI-H2444 CTRP2 7.365 17.3138 1.4689 16.022
NCI-H1838 CTRP2 7.3851 9.3009 5.3511 1.1306
RERF-LC-Sq1 GDSC1 7.4165 14.8864 1.3422 12.7769
Lu-99A GDSC1 7.4222 15.8769 0.879 15.1496
LCLC-97TM1 CTRP2 7.4568 10.1638 5.0088 2.2649
NCI-H2228 CTRP2 7.5111 9.7353 5.2304 1.4225
SK-LU-1 CTRP2 7.5356 10.8393 4.7464 3.1599
NCI-H1395 CTRP2 7.5665 9.6344 5.303 1.1349
HCC4006 CTRP2 7.6218 9.0996 5.5467 0.41
NCI-H1373 CTRP2 7.7248 10.1141 5.1805 1.4002
HCC1195 CTRP2 7.7867 9.256 5.5566 0.3175
HCC78 CTRP2 7.8109 12.4849 4.1505 5.1215
NCI-H2291 CTRP2 7.8238 9.4911 5.4829 0.4627
NCI-H2286 CTRP2 7.8448 9.322 5.5557 0.2976
HCC2108 CTRP2 7.8467 9.3733 5.5373 0.3335
COR-L88 CTRP2 7.8711 9.8182 5.3755 0.7073
IA-LM CTRP2 7.9209 9.5786 5.4907 0.4014
NCI-H2009 CTRP2 7.97 9.5861 5.5082 0.345
NCI-H1792 GDSC1 8.0331 16.2594 1.0896 12.7643
NCI-H1755 CTRP2 8.0392 9.7889 5.4605 0.4165
NCI-H1793 GDSC1 8.0703 20.361 -0.8296 20.817
NCI-H441 CTRP2 8.1125 9.7012 5.5228 0.2682
NCI-H1339 CTRP2 8.209 9.6214 5.5878 0.1452
NCI-H2085 CTRP2 8.2254 10.203 5.3815 0.5092
NCI-H2030 CTRP2 8.2568 9.8682 5.5183 0.2336
NCI-H2172 CTRP2 8.2923 10.2272 5.4004 0.44
NCI-H835 GDSC1 8.3828 22.1665 -1.4847 22.3085
LXF 289 GDSC1 8.4438 18.7961 0.164 16.1926
HCC1171 CTRP2 8.5564 10.2072 5.5105 0.1737
NCI-H1105 GDSC1 8.6155 23.4741 -1.9551 23.2292
COR-L105 GDSC1 8.7577 17.0032 1.1854 10.8709
NCI-H1869 GDSC1 9.176 22.0756 -0.9087 18.8402
RERF-LC-MS GDSC1 9.549 20.859 -0.1028 15.1429
NCI-H292 CTRP2 9.6464 19.7902 1.8919 11.0626
NCI-H1623 GDSC1 9.6793 21.8854 -0.4978 16.4226
NCI-H460 CTRP2 10.0563 21.1135 1.5338 11.714
NCI-H1944 CTRP2 10.7007 32.8752 -3.716 23.912
NCI-H2122 CTRP2 11.17 22.6467 1.5266 10.3482
Hs 888.Lu CTRP2 6.6179 8.5976 5.2083 2.5496
⏷ Show the Full List of 306 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Lymphoma Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
CBTCi002-A GDSC1 5.0442 9.6379 2.2392 13.5884
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Thigh Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
H-STS CTRP2 3.6186 7.2997 2.973 18.5112
SYO-1 CTRP2 6.5632 11.5199 3.726 8.7732
Cancer Drug Sensitivity Data Curated from 70 Cell Line(s) in Ovary Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
2004 CTRP2 6.4379 10.421 4.1747 7.1292
A2780 CTRP2 2.9342 5.5774 2.7653 21.3022
A2780 GDSC1 3.1644 5.8594 2.4583 19.4505
TOV-112D GDSC1 4.1579 8.5464 2.0715 17.8628
COV434 CTRP2 4.6955 6.5638 4.4037 10.0416
ES-2 GDSC1 5.1557 7.2549 3.4785 4.1681
DOV13 GDSC1 5.2884 8.5459 2.951 7.7287
TYK-nu CTRP2 5.294 7.691 4.5349 7.9592
TYK-nu GDSC1 5.3789 12.0143 1.3172 18.2985
OVCAR-3 GDSC1 5.4011 7.3937 3.5649 3.0104
Caov-3 GDSC1 5.4104 7.2525 3.6335 2.5295
OV7 CTRP2 5.4475 7.9561 4.5548 7.5172
OC 314 CTRP2 5.4636 8.118 4.4911 7.7437
DOV13 CTRP2 5.4795 12.4724 2.3483 16.4367
SK-OV-3 GDSC1 5.4795 9.2287 2.7534 8.6542
FU-OV-1 GDSC1 5.5884 9.4812 2.7062 8.702
RMG-I GDSC1 5.6046 8.4897 3.1853 5.2309
OVISE GDSC1 5.6586 7.7116 3.5687 2.5042
OVCAR-4 GDSC1 5.6595 8.933 3.013 6.3297
JHOS-2 GDSC1 5.6794 8.4497 3.2497 4.6115
OVCAR-5 CTRP2 5.7909 6.7686 5.4542 3.0178
JHOS-4 GDSC1 5.8398 13.3734 0.9904 18.6723
OAW42 CTRP2 5.8612 6.9027 5.4544 2.8577
TOV-21G GDSC1 5.8662 11.1216 2.1071 12.0561
SNU-119 CTRP2 5.9396 7.6981 5.1287 4.0563
EFO-27 GDSC1 5.965 11.1184 2.1763 11.3389
IGROV-1 GDSC1 6.0325 11.1681 2.1981 11.0193
Caov-4 GDSC1 6.0988 9.8858 2.8444 6.498
Kuramochi GDSC1 6.1276 11.3762 2.1624 11.0071
TOV-21G CTRP2 6.1671 7.6496 5.3416 2.7255
OAW28 GDSC1 6.1693 10.1696 2.7567 6.9383
OC 314 GDSC1 6.2088 8.115 3.6726 1.167
JHOC-5 CTRP2 6.2163 9.0947 4.66 5.4955
COV644 CTRP2 6.2215 7.6118 5.403 2.3729
Caov-3 CTRP2 6.2266 8.8042 4.8133 4.8338
EFO-21 GDSC1 6.279 8.7775 3.4363 2.3369
COV362 CTRP2 6.3246 7.7801 5.3976 2.2234
OVCAR-5 GDSC1 6.3306 8.1879 3.6976 0.9387
OVTOKO GDSC1 6.3965 10.0199 2.9597 5.1107
HEY A8 CTRP2 6.457 9.8856 4.4558 5.9217
ES2 CTRP2 6.4764 12.5954 3.1216 11.4046
OV56 CTRP2 6.543 8.3169 5.2921 2.3195
TOV-112D CTRP2 6.6064 15.8161 1.6186 16.8748
OV-90 CTRP2 6.6191 8.9712 5.0279 3.2828
OAW28 CTRP2 6.6387 8.6768 5.1845 2.6155
JHOS-2 CTRP2 6.6743 8.2491 5.4124 1.6584
OVK18 CTRP2 6.6756 8.7379 5.1805 2.5787
SNU-8 CTRP2 6.7124 11.1473 4.026 7.2731
RMG-I CTRP2 6.7689 8.9458 5.144 2.5934
OVCAR-8 GDSC1 6.812 11.585 2.4959 7.2774
JHOM-1 CTRP2 6.8196 8.3496 5.4559 1.3175
MCAS CTRP2 6.8986 17.0746 1.224 17.6843
EFO-27 CTRP2 6.9075 8.5987 5.3947 1.4463
OVKATE GDSC1 6.9083 8.2407 3.8973 0.1058
OAW42 GDSC1 6.9137 12.5835 2.0993 9.5389
OVTOKO CTRP2 6.9706 10.2557 4.6517 4.2892
OV-90 GDSC1 7.0509 13.121 1.9353 10.2282
OVSAHO CTRP2 7.0731 9.916 4.8842 3.2119
SK-OV-3 CTRP2 7.0812 8.5329 5.521 0.8324
OVCAR-4 CTRP2 7.1097 10.5576 4.602 4.2884
IGROV-1 CTRP2 7.1486 15.4283 2.2379 13.6452
Kuramochi CTRP2 7.2206 9.1668 5.3202 1.3872
SNU-840 CTRP2 7.2247 9.1318 5.3379 1.3213
OVK18 GDSC1 7.254 8.7483 3.846 0.1133
OV56 GDSC1 7.4318 13.7009 1.9009 9.6187
ONCO-DG-1 CTRP2 7.5427 18.2315 1.15 16.7857
EFO-21 CTRP2 7.7535 9.2539 5.5437 0.358
FU-OV-1 CTRP2 8.0275 10.3696 5.2257 1.027
OVCAR-8 CTRP2 10.4334 19.6422 2.4618 8.1269
OVISE CTRP2 13.4779 28.04 0.4505 10.9814
⏷ Show the Full List of 70 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 44 Cell Line(s) in Soft Tissue Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
Aska-SS CTRP2 6.8587 10.804 4.3044 5.8826
Yamato-SS CTRP2 7.2597 10.3307 4.8097 3.2593
A-204 CTRP2 3.6004 6.3673 3.2825 17.4074
A-204 GDSC1 3.9474 9.2927 1.5179 22.2136
KYM-1 GDSC1 4.0553 9.8784 1.3185 22.9269
EW-8 GDSC1 4.1238 7.9697 2.3304 16.1865
Rh30 GDSC1 4.5132 9.8851 1.6981 18.9579
SW982 CTRP2 4.6598 7.3173 4.064 11.4512
Rh41 CTRP2 4.683 7.0353 4.2065 10.8324
TTC-709 CTRP2 4.6924 8.0199 3.7863 12.4689
G-401 GDSC1 4.7237 10.0883 1.7664 17.7839
Hs 633.T GDSC1 4.8187 6.3941 3.6649 3.6343
G-402 CTRP2 4.8607 7.2153 4.3158 9.9293
SW872 GDSC1 4.992 6.7952 3.5892 3.7547
G-402 GDSC1 5.0349 10.0454 2.0305 15.031
SK-LMS-1 GDSC1 5.0553 9.9068 2.1147 14.4023
MFH-ino GDSC1 5.1584 10.7325 1.7842 16.2227
SW684 GDSC1 5.1914 7.9554 3.1687 6.3728
VA-ES-BJ GDSC1 5.337 7.5977 3.4329 4.0735
G-401 CTRP2 5.5546 8.1497 4.5601 7.2537
GCT GDSC1 5.622 9.8898 2.5328 9.8374
Rh41 GDSC1 5.6794 10.8039 2.1307 12.4179
HT-1080 GDSC1 5.8196 10.794 2.233 11.3524
HT-1080 CTRP2 5.8305 6.7725 5.4897 2.7802
TE 617.T CTRP2 6.0201 7.1768 5.4578 2.5129
TE 441.T CTRP2 6.0567 6.9342 5.6097 1.8037
Hs 729.T CTRP2 6.0592 8.7722 4.6928 5.6524
SW982 GDSC1 6.1537 7.651 3.8268 0.5605
Rh18 CTRP2 6.1665 8.479 4.9273 4.4652
SK-UT-1 GDSC1 6.2995 9.9702 2.926 5.5238
KYM-1 CTRP2 6.3504 9.4916 4.5687 5.637
Rh18 GDSC1 6.3585 10.3144 2.8047 6.208
RKN GDSC1 6.4193 7.8193 3.8685 0.2909
RKN CTRP2 6.4596 7.9937 5.3903 2.0439
SK-LMS-1 CTRP2 6.4624 9.1748 4.8125 4.4252
RD CTRP2 6.4695 9.5651 4.6246 5.196
SK-UT-1 CTRP2 6.4772 9.8371 4.4956 5.7209
GCT CTRP2 6.5097 8.3076 5.2732 2.4462
BT-16 CTRP2 6.7354 15.9382 1.6608 16.4852
MES-SA GDSC1 6.9918 13.1471 1.8863 10.6515
BT-12 CTRP2 7.2411 11.216 4.3752 5.0137
Tm87-16 CTRP2 7.6569 10.5658 4.9441 2.2856
MES-SA CTRP2 7.9361 9.2268 5.6256 0.1533
RD GDSC1 8.9338 18.9744 0.3894 14.2465
⏷ Show the Full List of 44 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Clivus Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
U-CH1 CTRP2 7.7673 9.3106 5.528 0.3862
Cancer Drug Sensitivity Data Curated from 14 Cell Line(s) in Pleura Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
MSTO-211H GDSC1 4.4093 8.9688 2.0709 16.9178
MSTO-211H CTRP2 5.1302 7.0142 4.6809 7.7808
MPP 89 GDSC1 5.5364 12.7598 1.0674 19.1719
NCI-H2452 GDSC1 5.8707 10.3241 2.4927 9.4603
NCI-H2052 GDSC1 5.981 8.9062 3.2203 4.1948
NCI-H28 GDSC1 6.0321 11.5723 2.004 12.2741
ACC-MESO-1 CTRP2 6.2016 11.0184 3.6871 9.5947
NCI-H28 CTRP2 6.546 8.7839 5.0668 3.2363
MPP 89 CTRP2 6.6745 8.9275 5.0882 2.9535
IST-Mes1 CTRP2 6.688 11.1667 3.9978 7.4311
NCI-H2052 CTRP2 7.9491 11.2379 4.8107 2.4623
NCI-H2452 CTRP2 8.0462 10.0575 5.3599 0.6488
IST-Mes1 GDSC1 8.2819 17.6985 0.5755 14.7161
JL-1 CTRP2 15.299 44.6456 -6.1944 22.6834
⏷ Show the Full List of 14 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 10 Cell Line(s) in Prostate Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
PC-3 GDSC1 5.2139 9.3384 2.5126 11.141
VCaP GDSC1 5.2937 9.2802 2.5986 10.2889
LNCaP clone FGC CTRP2 5.6662 8.5957 4.4413 7.5057
22Rv1 GDSC1 5.6735 8.7333 3.1151 5.5715
DU145 CTRP2 6.188 7.9222 5.2223 3.188
LNCaP clone FGC GDSC1 6.3358 14.2675 0.9112 17.6917
VCaP CTRP2 6.4379 7.8826 5.429 1.9187
PaCa-3 CTRP2 6.9063 8.37 5.4971 1.0754
22Rv1 CTRP2 7.0205 9.4808 5.0557 2.6063
DU145 GDSC1 9.0854 19.5835 0.2011 14.764
⏷ Show the Full List of 10 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 2 Cell Line(s) in Salivary Gland Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
A-253 GDSC1 5.8862 8.8097 3.2088 4.4606
YD-15 CTRP2 6.2561 8.512 4.9822 4.0725
Cancer Drug Sensitivity Data Curated from 1 Cell Line(s) in Small Intestine Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HuTu 80 GDSC1 5.1337 9.578 2.336 12.6349
Cancer Drug Sensitivity Data Curated from 58 Cell Line(s) in Stomach Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
HSC-39 GDSC1 -0.7594 3.8373 -1.0991 59.9364
KATO III GDSC1 0.4275 3.9902 0.1576 48.8869
SNU-16 CTRP2 2.602 4.7223 2.549 23.1125
GSS CTRP2 3.7262 7.2827 3.0943 17.7487
SNU-1 CTRP2 4.0037 6.8698 3.5478 15.2456
ECC10 GDSC1 4.6164 11.9038 0.7735 23.6687
HGC-27 CTRP2 4.6905 7.1767 4.1555 11.0106
SNU-1 GDSC1 4.8363 9.3714 2.212 14.4544
SNU-620 CTRP2 4.8725 7.0029 4.4185 9.4948
OCUM-1 GDSC1 5.2376 10.0239 2.1934 13.2971
Fu97 GDSC1 5.2599 9.0235 2.6996 9.6557
ECC10 CTRP2 5.2703 6.3252 5.1092 5.7385
AGS GDSC1 5.288 11.7769 1.3657 18.3101
MKN28 GDSC1 5.3979 8.17 3.2037 5.587
MKN45 GDSC1 5.4772 6.404 4.0161 0.3303
IM95 GDSC1 5.4789 7.915 3.3735 4.1786
MKN7 GDSC1 5.5121 8.571 3.0886 6.1432
RF-48 GDSC1 5.5333 7.659 3.5221 3.0401
23132/87 CTRP2 5.5334 9.7458 3.7523 10.6617
23132/87 GDSC1 5.5893 7.9292 3.433 3.5332
SNU-601 CTRP2 5.635 8.0266 4.6944 6.5174
Hs 746.T GDSC1 5.6671 8.8484 3.0574 5.9957
TGBC11TKB GDSC1 5.7029 12.0567 1.5364 16.0613
KATO III CTRP2 5.787 15.9459 0.8776 20.9782
SCH GDSC1 5.8466 7.3046 3.8295 0.7942
KE-39 CTRP2 5.8627 8.6446 4.59 6.4732
NUGC-4 GDSC1 5.8921 11.0351 2.1667 11.5962
Hs 746.T CTRP2 5.946 7.385 5.2904 3.3644
IM95 CTRP2 5.9517 8.6358 4.6706 5.9558
MKN1 GDSC1 5.9876 7.8764 3.6663 1.4458
SNU-16 GDSC1 6.0269 7.3033 3.904 0.3759
MKN1 CTRP2 6.1236 8.0091 5.1272 3.7052
HGC-27 GDSC1 6.1257 7.6802 3.8044 0.6653
GSU CTRP2 6.1905 7.8243 5.273 2.9711
NUGC-4 CTRP2 6.3576 9.0629 4.7875 4.7086
SNU-5 GDSC1 6.4334 7.7266 3.9058 0.2009
NUGC-3 CTRP2 6.467 8.8597 4.9715 3.7568
SNU-668 CTRP2 6.4977 7.9966 5.4154 1.8866
NCI-N87 GDSC1 6.5028 8.6945 3.576 1.3268
NUGC-3 GDSC1 6.5579 8.0077 3.8535 0.2738
SNU-216 CTRP2 6.6176 9.6672 4.6857 4.6955
GCIY GDSC1 6.6939 8.5221 3.7215 0.5844
NCI-N87 CTRP2 6.8014 8.5842 5.3363 1.7933
SNU-719 CTRP2 6.8586 8.6465 5.3431 1.6972
ECC12 CTRP2 7.0679 11.1796 4.2718 5.69
LMSU CTRP2 7.1227 10.982 4.4062 5.0608
MKN7 CTRP2 7.1549 8.737 5.4722 0.9298
RERF-GC-1B GDSC1 7.2903 11.5961 2.7592 4.7773
MKN74 CTRP2 7.5516 10.2527 5.024 2.1075
HuG1-N CTRP2 7.7081 9.715 5.3402 0.9125
MKN45 CTRP2 8.0853 20.799 0.2912 18.5453
Fu97 CTRP2 8.2415 9.8624 5.5145 0.2439
AGS CTRP2 8.6012 14.4267 3.7441 5.6812
SH-10-TC CTRP2 10.0236 20.4898 1.8078 10.849
SNG-M GDSC1 4.0126 7.5209 2.4579 15.7005
SNU-1077 CTRP2 4.8958 6.7232 4.5571 8.8942
SNU-685 CTRP2 7.1326 9.1715 5.2676 1.6672
SNG-M CTRP2 12.0767 25.9136 0.5741 12.1661
⏷ Show the Full List of 58 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 28 Cell Line(s) in Thyroid Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
IHH-4 GDSC1 3.1947 9.6947 0.6466 29.8882
8505C GDSC1 3.4833 14.3493 -1.4067 35.2632
CGTH-W-1 CTRP2 3.9793 6.8986 3.5109 15.4543
SW579 CTRP2 4.7165 7.0289 4.2442 10.5948
CGTH-W-1 GDSC1 4.8406 10.7053 1.5515 18.6981
CAL-62 CTRP2 5.029 8.0088 4.1261 10.2636
CAL-62 GDSC1 5.4397 12.6965 1.0258 19.686
FTC-133 GDSC1 5.4489 7.0855 3.7278 1.8532
B-CPAP GDSC1 5.4498 7.1899 3.683 2.1352
ML-1 [Human leukemia] GDSC1 5.6695 11.7949 1.6403 15.5421
ASH-3 GDSC1 5.7899 12.1654 1.5461 15.7517
FTC-238 CTRP2 5.8031 7.0916 5.3082 3.5938
8505C CTRP2 5.8039 9.6876 4.0187 8.9876
8305C GDSC1 6.1588 7.7045 3.8089 0.6233
K5 GDSC1 6.1646 8.7122 3.4056 2.6887
WRO GDSC1 6.1799 7.9003 3.7435 0.8723
B-CPAP CTRP2 6.392 10.2771 4.2103 7.062
BHT-101 GDSC1 6.5137 14.4668 0.9396 17.0752
TT CTRP2 6.5165 9.0863 4.8967 3.986
KMH-2 GDSC1 6.6043 8.116 3.8327 0.3063
TT GDSC1 6.6046 7.9705 3.8832 0.1951
FTC-133 CTRP2 6.6769 9.1073 5.0027 3.2983
BHT-101 CTRP2 6.7142 9.569 4.8043 4.053
TT2609-C02 GDSC1 6.7608 10.2083 3.0768 3.7347
8305C CTRP2 6.787 9.4263 4.9252 3.4499
HTC-C3 GDSC1 6.7969 9.1275 3.5365 1.2264
TT2609-C02 CTRP2 6.9316 8.7417 5.3438 1.6089
ML-1 [Human leukemia] CTRP2 7.0245 8.9476 5.3055 1.6467
⏷ Show the Full List of 28 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 68 Cell Line(s) in Upper Aerodigestive Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
YD-10B CTRP2 4.5998 7.714 3.8297 12.5328
NCI-H3118 GDSC1 4.6818 7.3817 3.0806 8.5442
PCI-04B GDSC1 5.1327 12.1637 1.0545 20.5077
BICR 22 GDSC1 5.2182 7.87 3.2278 5.8624
HO-1-u-1 GDSC1 5.2477 8.3699 3.0079 7.4187
CAL-33 CTRP2 5.3884 8.5881 4.1916 9.1537
HSC-2 CTRP2 5.425 6.6943 5.1238 5.2592
CAL-27 GDSC1 5.4463 7.7056 3.45 3.7122
BB30-HNC GDSC1 5.4519 7.7723 3.4227 3.8912
Ca9-22 GDSC1 5.4819 8.1274 3.2771 4.8575
OSC-20 GDSC1 5.4986 11.4023 1.7081 15.6385
PCI-30 GDSC1 5.6214 7.5807 3.6056 2.333
KOSC-2 GDSC1 5.6733 11.3778 1.847 14.2622
PE/CA-PJ15 GDSC1 5.7318 9.4851 2.7995 7.6713
OSC-19 GDSC1 5.8055 8.0794 3.488 2.7653
SAT [Human HNSCC] GDSC1 5.8384 10.4805 2.3964 10.2022
FaDu CTRP2 5.8666 9.1248 4.3536 7.4573
CAL-33 GDSC1 5.874 10.0032 2.6473 8.3853
BHY GDSC1 5.8823 9.1268 3.0618 5.4778
HO-1-N-1 GDSC1 5.9704 8.9989 3.1725 4.5364
SCC-4 GDSC1 5.9871 10.8378 2.3254 10.2938
SCC-15 GDSC1 6.0253 8.0428 3.6163 1.6679
SNU-1214 CTRP2 6.1672 7.4521 5.4401 2.3128
BICR 78 GDSC1 6.188 8.4836 3.5137 2.0226
HSC-2 GDSC1 6.2039 7.7694 3.8031 0.6131
HSC-3 GDSC1 6.2478 7.6614 3.8601 0.3933
KON GDSC1 6.2835 7.7278 3.8499 0.4056
HSC-4 CTRP2 6.2886 9.7189 4.4065 6.4271
BICR 18 CTRP2 6.3773 7.9067 5.374 2.2367
PCI-15A GDSC1 6.4388 8.053 3.7924 0.5008
PE/CA-PJ49 CTRP2 6.4505 7.7576 5.4981 1.6208
PE/CA-PJ15 CTRP2 6.4515 9.4277 4.6789 5.0001
BICR 31 GDSC1 6.4673 11.8245 2.1724 10.1039
Detroit 562 GDSC1 6.4971 8.074 3.8073 0.423
PCI-38 GDSC1 6.5041 8.3476 3.7098 0.7509
SNU-1076 CTRP2 6.5162 19.6146 -0.3517 23.1346
PE/CA-PJ34 (clone C12) CTRP2 6.553 9.1293 4.9025 3.9028
LB771-HNC GDSC1 6.5571 8.8293 3.5472 1.4085
FaDu GDSC1 6.5776 7.8317 3.9208 0.1358
CAL-27 CTRP2 6.6206 9.9496 4.5487 5.2581
PE/CA-PJ41 (clone D2) CTRP2 6.6255 8.0705 5.465 1.5157
YD-8 CTRP2 6.6279 8.4258 5.2979 2.1743
SCC-9 GDSC1 6.6518 8.1126 3.8512 0.2462
SNU-46 CTRP2 6.6576 9.0013 5.0405 3.1728
JHU-022 GDSC1 6.7607 8.8761 3.6171 0.9193
SAS GDSC1 6.7733 8.5058 3.758 0.4305
BICR 10 GDSC1 6.7764 8.1908 3.8687 0.1758
SCC-25 GDSC1 6.8142 8.7159 3.698 0.5911
DOK GDSC1 6.8209 12.2648 2.1895 9.1863
HSC-4 GDSC1 6.8812 8.2455 3.8865 0.1249
BB49-HNC GDSC1 6.8954 8.8008 3.6988 0.5435
SNU-899 CTRP2 6.958 9.048 5.2185 2.0536
BHY CTRP2 6.9761 11.3253 4.1344 6.3947
BICR 16 CTRP2 6.9865 9.9653 4.8027 3.6567
JHU-011 GDSC1 6.9895 14.3738 1.3075 13.9499
SNU-1066 CTRP2 7.0448 9.8362 4.9034 3.174
BICR 22 CTRP2 7.0635 10.7983 4.4539 4.9551
SCC-25 CTRP2 7.216 8.8982 5.435 0.9995
SKN-3 GDSC1 7.2314 9.2099 3.6802 0.4361
BICR 6 CTRP2 7.2941 21.5501 -0.6932 22.6086
SCC-9 CTRP2 7.4637 10.2166 4.9888 2.3308
PCI-06A GDSC1 7.5713 15.1746 1.3055 12.6312
SNU-1041 CTRP2 7.8063 10.4255 5.0894 1.6316
Detroit 562 CTRP2 7.9175 11.6048 4.6267 3.167
HSC-3 CTRP2 7.9644 13.2302 3.898 5.9059
BICR 56 CTRP2 8.1702 9.7188 5.5388 0.2245
SCC-4 CTRP2 8.2581 9.7963 5.5445 0.1934
BICR 31 CTRP2 8.3858 10.1183 5.4779 0.2629
⏷ Show the Full List of 68 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 39 Cell Line(s) in Urinary Tract Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
JMSU-1 CTRP2 2.8509 7.4729 2.0864 24.0016
639V GDSC1 4.1031 6.7339 2.929 11.7817
RT-4 GDSC1 4.6312 10.2715 1.6008 19.13
RT-112 GDSC1 4.8579 9.2278 2.3001 13.769
RT-112 CTRP2 4.9451 8.9656 3.5903 12.6473
KU-19-19 GDSC1 5.2208 8.3188 3.0139 7.4471
BFTC-905 GDSC1 5.3288 11.0806 1.7406 15.9575
253J CTRP2 5.3299 8.5542 4.1537 9.4425
UM-UC-3 GDSC1 5.4422 7.6638 3.4666 3.6047
5637 GDSC1 5.4558 9.1822 2.7596 8.6735
HT-1197 CTRP2 5.5299 6.5726 5.2848 4.3483
5637 CTRP2 5.6353 8.2161 4.6013 6.9046
SW780 GDSC1 5.6685 10.286 2.3738 10.8124
SW1710 GDSC1 5.6893 9.4521 2.7873 7.8646
T24 GDSC1 5.7211 9.6924 2.6941 8.4431
UM-UC-3 CTRP2 5.7266 7.2521 5.1589 4.3846
UM-UC-1 CTRP2 5.8298 15.7879 0.9926 20.5198
647V GDSC1 5.8317 9.1526 3.0188 5.889
HT-1376 GDSC1 5.8574 8.7685 3.2105 4.5079
647V CTRP2 5.8704 8.408 4.7146 5.9346
TCCSUP CTRP2 6.1219 8.3124 4.9743 4.3507
BC-3C CTRP2 6.136 7.6026 5.3403 2.7876
RT-4 CTRP2 6.1462 8.5848 4.858 4.7941
CAL-29 GDSC1 6.2205 7.9744 3.7324 0.8846
U-BLC1 CTRP2 6.3369 7.5816 5.5039 1.7659
HT-1197 GDSC1 6.3416 7.9264 3.8004 0.5322
VM-CUB-1 CTRP2 6.3742 8.644 5.0082 3.7592
J82 CTRP2 6.3846 8.5574 5.0589 3.5304
KMBC-2 CTRP2 6.3883 7.7777 5.4449 1.9286
CAL-29 CTRP2 6.4746 9.2057 4.8064 4.4302
BFTC-905 CTRP2 6.4893 8.1402 5.3401 2.2039
SCaBER CTRP2 6.501 8.8646 4.9944 3.6067
J82 GDSC1 6.5233 10.8323 2.6669 6.7723
639V CTRP2 6.8223 11.1531 4.1058 6.7603
T24 CTRP2 6.8687 11.8595 3.792 7.9768
HT-1376 CTRP2 7.1585 11.0069 4.4191 4.9562
TCCSUP GDSC1 7.6351 15.6291 1.1333 13.39
SW1710 CTRP2 7.6678 16.7527 1.9756 13.7246
KU-19-19 CTRP2 10.0696 25.0894 -0.3678 17.3756
⏷ Show the Full List of 39 Cancer Drug Sensitivity Data of This Drug
Cancer Drug Sensitivity Data Curated from 40 Cell Line(s) in Urogenital System Tissue
Cell Line Original Dataset IC50 IC90 EC50 AUC
NEC8 GDSC1 2.94 6.3131 2.0266 23.564
HEY GDSC1 3.711 8.0092 1.9473 20.5108
SKN GDSC1 4.5815 6.3202 3.53 5.366
TC-YIK GDSC1 4.5908 9.143 2.1317 15.8502
Ca Ski GDSC1 4.6486 9.2856 2.1068 15.8172
NCC-IT GDSC1 4.7686 6.7546 3.4548 5.3803
PA-1 GDSC1 5.1496 7.5111 3.3532 5.1074
SW962 GDSC1 5.2158 9.7937 2.2905 12.6984
BPH-1 GDSC1 5.2245 7.8125 3.2594 5.612
JAR GDSC1 5.346 9.0666 2.7394 9.1218
LB831-BLC GDSC1 5.3952 9.0678 2.773 8.7417
C-33 A GDSC1 5.4053 8.9774 2.8235 8.3468
KGN GDSC1 5.4375 8.9791 2.8447 8.106
NT2-D1 GDSC1 5.4746 10.2356 2.262 12.1235
OVCA433 GDSC1 5.4806 8.2241 3.2313 5.1892
PWR-1E GDSC1 5.5371 12.9619 0.9681 19.6865
C-4-I GDSC1 5.5894 10.7109 2.1123 12.796
OMC-1 [Human cervical carcinoma] GDSC1 5.5906 9.2804 2.8036 7.9999
HeLa GDSC1 5.6512 7.2897 3.7448 1.4493
PEO1 GDSC1 5.7196 9.3561 2.8526 7.3255
HEC-1 GDSC1 5.7364 8.2016 3.3955 3.4968
SiHa GDSC1 5.7628 11.3748 1.9122 13.5956
CAL-39 GDSC1 5.8011 10.2174 2.4972 9.6098
DSH1 GDSC1 5.853 8.1586 3.4793 2.7396
SW954 GDSC1 5.9353 10.5702 2.4185 9.8008
OVCA420 GDSC1 6.0592 8.2079 3.5647 1.9104
ACC-OV7 GDSC1 6.0617 8.6383 3.3831 2.9928
JEG-3 GDSC1 6.0633 12.231 1.7078 14.0241
ME-180 GDSC1 6.1143 11.1211 2.275 10.3048
SW756 GDSC1 6.3747 7.7748 3.8677 0.3115
UWB1.289 GDSC1 6.55 11.6872 2.2891 9.1657
MS751 GDSC1 6.5869 8.0862 3.8367 0.3032
SiSo GDSC1 6.6942 8.7989 3.6185 0.9659
JHOS-3 GDSC1 6.8256 8.8022 3.671 0.6747
DoTc2 4510 GDSC1 6.9822 8.719 3.7605 0.3356
OV17R GDSC1 7.006 9.2486 3.5783 0.8877
SKG-IIIa GDSC1 7.0862 8.5311 3.8612 0.1219
HT-3 GDSC1 7.3055 8.7914 3.8491 0.102
OVMIU GDSC1 7.6428 9.8732 3.5992 0.4724
HeLa CTRP2 8.5492 28.763 -3.3009 26.1932
⏷ Show the Full List of 40 Cancer Drug Sensitivity Data of This Drug

References

1 URL: http://www.guidetopharmacology.org Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 5671).
2 Interpreting expression profiles of cancers by genome-wide survey of breadth of expression in normal tissues. Genomics 2005 Aug;86(2):127-41.